MECHANISMS OF NONCOMPETITIVE INHIBITION OF ACETYLCHOLINE-INDUCED SINGLE-CHANNEL CURRENTS

被引:62
作者
PAPKE, RL [1 ]
OSWALD, RE [1 ]
机构
[1] CORNELL UNIV,COLL VET MED,DEPT PHARMACOL,ITHACA,NY 14853
关键词
D O I
10.1085/jgp.93.5.785
中图分类号
Q4 [生理学];
学科分类号
071003 ;
摘要
引用
收藏
页码:785 / 811
页数:27
相关论文
共 44 条
[1]  
AGUAYO LG, 1981, MOL PHARMACOL, V20, P345
[2]   VOLTAGE-DEPENDENT AND TIME-DEPENDENT EFFECTS OF PHENCYCLIDINES ON THE END-PLATE CURRENT ARISE FROM OPEN AND CLOSED CHANNEL BLOCKADE [J].
AGUAYO, LG ;
WITKOP, B ;
ALBUQUERQUE, EX .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (10) :3523-3527
[3]  
ARACAVA Y, 1984, MOL PHARMACOL, V26, P303
[4]   QUATERNARY STRUCTURE OF THE ACETYLCHOLINE-RECEPTOR [J].
BRISSON, A ;
UNWIN, PNT .
NATURE, 1985, 315 (6019) :474-477
[5]  
CACECI MS, 1984, BYTE, V9, P340
[6]   ELECTRO-PHYSIOLOGICAL AND BIOCHEMICAL-STUDIES ON ENHANCEMENT OF DESENSITIZATION BY PHENOTHIAZINE NEUROLEPTICS [J].
CARP, JS ;
ARONSTAM, RS ;
WITKOP, B ;
ALBUQUERQUE, EX .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (01) :310-314
[7]   EFFECTS OF CHLORPROMAZINE AND PHENCYCLIDINE ON MOUSE C2 ACETYLCHOLINE-RECEPTOR KINETICS [J].
CHANGEUX, JP ;
PINSET, C ;
RIBERA, AB .
JOURNAL OF PHYSIOLOGY-LONDON, 1986, 378 :497-513
[8]  
CHANGEUX JP, 1981, HARVEY LECT, V75, P85
[9]  
COHEN JB, 1980, PSYCHOPHARMACOLOGY B, P47
[10]  
COLEMAN BA, 1987, MOL PHARMACOL, V32, P456