A DIRECT ROUTE TO THE PYRROLO[2,1-C][1,4]BENZODIAZEPINE RING-SYSTEM USING ARYL TRIFLATES

被引：23

作者：

KRAUS, GA

LIU, P

机构：

[1] Department of Chemistry, Iowa State University, Ames

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 42期

关键词：

TRIFLATE; BENZODIAZEPINE; ANTIBIOTICS;

D O I：

10.1016/0040-4039(95)01592-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The pyrrolo[2,1-c][1,4]benzodiazepine and dibenzo[b,e][1,4] diazepine skeletons were rapidly generated from salicylic acids. The key step in these syntheses was the substitution of an aryl triflate.

引用

页码：7595 / 7598

页数：4

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