A STEREOSPECIFIC SYNTHESIS OF A RENIN INHIBITOR (BW-175) WHICH INCORPORATES A SULFONEMETHYLENE ISOSTERE AND A DIHYDROXYETHYLENE ISOSTERE

被引：14

作者：

NAKANO, M

ATSUUMI, S

KOIKE, Y

TANAKA, S

FUNABASHI, H

HASHIMOTO, J

MORISHIMA, H

机构：

[1] Chemistry of Natural Products, Exploratory Research Laboratories, Banyu Pharmaceutical CO., Meguro-ku, Tokyo, 153, 2-9-3, Shimomeguro

来源：

TETRAHEDRON LETTERS | 1990年 / 31卷 / 11期

关键词：

D O I：

10.1016/0040-4039(90)80019-I

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1569 / 1572

页数：4

共 15 条

[1] CATALYTIC TRANSFER HYDROGENATION
BRIEGER, G
NESTRICK, TJ
[J]. CHEMICAL REVIEWS, 1974, 74 (05) : 567 - 580
[2] ASYMMETRIC-SYNTHESIS OF THE ENKEPHALINASE INHIBITOR THIORPHAN
EVANS, DA
MATHRE, DJ
SCOTT, WL
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1985, 50 (11) : 1830 - 1835
[3] CONTRASTERIC CARBOXIMIDE HYDROLYSIS WITH LITHIUM HYDROPEROXIDE
EVANS, DA
BRITTON, TC
ELLMAN, JA
[J]. TETRAHEDRON LETTERS, 1987, 28 (49) : 6141 - 6144
[4] ASYMMETRIC ALKYLATION REACTIONS OF CHIRAL IMIDE ENOLATES - A PRACTICAL APPROACH TO THE ENANTIOSELECTIVE SYNTHESIS OF ALPHA-SUBSTITUTED CARBOXYLIC-ACID DERIVATIVES
EVANS, DA
ENNIS, MD
MATHRE, DJ
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1982, 104 (06) : 1737 - 1739
[5] RENIN INHIBITORS
GREENLEE, WJ
[J]. PHARMACEUTICAL RESEARCH, 1987, 4 (05) : 364 - 374
[6] HANESSIAN S, 1981, SYNTHESIS-STUTTGART, P396
[7] SYNTHETIC AND ENZYME-INHIBITION STUDIES OF PEPSTATIN ANALOGS CONTAINING HYDROXYETHYLENE AND KETOMETHYLENE DIPEPTIDE ISOSTERES
HOLLADAY, MW
SALITURO, FG
RICH, DH
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (02) : 374 - 383
[8] RENIN INHIBITORS - IMPROVEMENTS IN THE STABILITY AND BIOLOGICAL-ACTIVITY OF SMALL PEPTIDES CONTAINING NOVEL LEU-VAL REPLACEMENTS
KLEINERT, HD
LULY, JR
MARCOTTE, PA
PERUN, TJ
PLATTNER, JJ
STEIN, H
[J]. FEBS LETTERS, 1988, 230 (1-2) : 38 - 42
[9] LAL B, 1977, TETRAHEDRON LETT, P1977
[10] THE USE OF DIETHYL AZODICARBOXYLATE AND TRIPHENYLPHOSPHINE IN SYNTHESIS AND TRANSFORMATION OF NATURAL-PRODUCTS
MITSUNOBU, O
[J]. SYNTHESIS-STUTTGART, 1981, (01): : 1 - 28

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