SYNTHESIS AND ANALGETIC ACTIVITY OF SOME 1-SUBSTITUTED 3-PYRROLIDINYLANILIDES AND DIHYDROBENZOXAZINONES

被引：17

作者：

HELSLEY, GC

LUNSFORD, CD

WELSTEAD, WJ

BOSWELL, RF

FUNDERBURK, WH

JOHNSON, DN

机构：

[1] Research Laboratories, A. H. Robins Company, Inc., Richmond, virginia

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1969年 / 12卷 / 04期

关键词：

D O I：

10.1021/jm00304a005

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Some 1-substituted 3-pyrrolidinylanilides and 1-substituted 3-pyrrolidinyl-2H-1,4-benzoxazin-3(4H)-ones have been prepared and tested for analgetic activity. Several of the compounds show moderate to potent activity. © 1969, American Chemical Society. All rights reserved.

引用

页码：583 / +

页数：1

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JOURNAL OF MEDICINAL CHEMISTRY, 1967, 10 (06) :1015-&

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