PRODRUGS OF TIMOLOL FOR IMPROVED OCULAR DELIVERY - SYNTHESIS, HYDROLYSIS KINETICS AND LIPOPHILICITY OF VARIOUS TIMOLOL ESTERS

被引：45

作者：

BUNDGAARD, H ^{[1
]}

BUUR, A ^{[1
]}

CHANG, SC ^{[1
]}

LEE, VHL ^{[1
]}

机构：

[1] UNIV SO CALIF,SCH PHARM,LOS ANGELES,CA 90089

来源：

INTERNATIONAL JOURNAL OF PHARMACEUTICS | 1986年 / 33卷 / 1-3期

关键词：

D O I：

10.1016/0378-5173(86)90034-7

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：15 / 26

页数：12

共 30 条

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[5] PILOCARPIC ACID-ESTERS AS NOVEL SEQUENTIALLY LABILE PILOCARPINE PRODRUGS FOR IMPROVED OCULAR DELIVERY
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[6] INTRAMOLECULAR AMINOLYSIS OF ESTERS - O-ACETYLSERINE AND GAMMA-ESTERS OF GLUTAMIC-ACID
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[9] ANALOGS OF NEUROEFFECTORS .V. NEIGHBORING-GROUP EFFECTS IN REACTIONS OF ESTERS THIOLESTERS AND SELENOLESTERS . HYDROLYSIS AND AMINOLYSIS OF BENZOYLCHOLINE BENZOYLTHIOLCHOLINE BENZOYLSELENOLCHOLINE AND OF THEIR DIMETHYLAMINO ANALOGS
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[10] BETA-ADRENERGIC BLOCKING AGENTS .2. PROPRANOLOL AND RELATED 3-AMINO-I-NAPHTHOXY-2-PROPANOLS
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