N,N-DIALLYL-TYROSYL SUBSTITUTION CONFERS ANTAGONIST PROPERTIES ON THE KAPPA-SELECTIVE OPIOID PEPTIDE [D-PRO10]DYNORPHIN A(1-11)

被引：24

作者：

GAIRIN, JE

MAZARGUIL, H

ALVINERIE, P

BOTANCH, C

CROS, J

MEUNIER, JC

机构：

来源：

BRITISH JOURNAL OF PHARMACOLOGY | 1988年 / 95卷 / 04期

关键词：

D O I：

10.1111/j.1476-5381.1988.tb11735.x

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：1023 / 1030

页数：8

共 22 条

[11] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF ANALOGS OF DYNORPHIN-A(1-13) SUBSTITUTED IN POSITION-2 AND POSITION-4 - DESIGN OF [ALA2,TRP4]-DYN-A(1-13) AS A PUTATIVE SELECTIVE OPIOID ANTAGONIST [J].

LEMAIRE, S ;

TURCOTTE, A .

CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1986, 64 (06) :673-678

[12] DESIGN AND USES OF SELECTIVE AGONISTIC AND ANTAGONISTIC ANALOGS OF THE NEUROPEPTIDES OXYTOCIN AND VASOPRESSIN [J].

MANNING, M ;

SAWYER, WH .

TRENDS IN NEUROSCIENCES, 1984, 7 (01) :6-9

[13] INCREASE IN POTENCIES OF OPIOID-PEPTIDES AFTER PEPTIDASE INHIBITION [J].

MCKNIGHT, AT ;

CORBETT, AD ;

KOSTERLITZ, HW .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 86 (3-4) :393-402

[14]

MEUNIER JC, 1983, MOL PHARMACOL, V24, P23

[15] RABBIT VAS-DEFERENS - A SPECIFIC BIOASSAY FOR OPIOID KAPPA-RECEPTOR AGONISTS [J].

OKA, T ;

NEGISHI, K ;

SUDA, M ;

MATSUMIYA, T ;

INAZU, T ;

UEKI, M .

EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 73 (2-3) :235-236

[16] CONTROL BY CATIONS OF OPIOID BINDING IN GUINEA-PIG BRAIN MEMBRANES [J].

PATERSON, SJ ;

ROBSON, LE ;

KOSTERLITZ, HW .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (16) :6216-6220

[17] AGONIST-ANTAGONIST PROPERTIES OF N-ALLYL-[D-ALA]2-MET-ENKEPHALIN [J].

PERT, CB ;

BOWIE, DL ;

PERT, A ;

MORELL, JL ;

GROSS, E .

NATURE, 1977, 269 (5623) :73-75

[18] TENA, A SELECTIVE KAPPA OPIOID RECEPTOR ANTAGONIST [J].

PORTOGHESE, PS ;

TAKEMORI, AE .

LIFE SCIENCES, 1985, 36 (08) :801-805

[19] BINALTORPHIMINE AND NOR-BINALTORPHIMINE, POTENT AND SELECTIVE KAPPA-OPIOID RECEPTOR ANTAGONISTS [J].

PORTOGHESE, PS ;

LIPKOWSKI, AW ;

TAKEMORI, AE .

LIFE SCIENCES, 1987, 40 (13) :1287-1292

[20] PEPTIDE ANTAGONISTS [J].

REGOLI, D .

TRENDS IN PHARMACOLOGICAL SCIENCES, 1985, 6 (12) :481-484

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