SYNTHESIS OF THE 3-AMINOFLAVONE-8-ACETIC ACID

被引：19

作者：

DAUZONNE, D

MARTINEZ, L

机构：

[1] Laboratoire de Chimie associé au CNRS, Institut Curie, Section de Biologie, 75231 Paris Cedex 05

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 11期

关键词：

D O I：

10.1016/0040-4039(95)00138-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of the so far unknown 3-amino-4-oxo-2-phenyl-4H-1-benzopyran-8-acetic acid (3-aminoflavone-8-acetic acid) starting from 2-hydroxy-3-(prop-2-ene)benzaldehyde and (Z)-(2-chloro-2-nitroethenyl)benzene is described.

引用

页码：1845 / 1848

页数：4

共 67 条

[1] SYNTHESIS AND ANTITUMOR-ACTIVITY OF 6-METHYL DERIVATIVES OF FLAVONE-8-ACETIC ACID (FAA) [J].

AITKEN, RA ;

BIBBY, MC ;

DOUBLE, JA ;

PHILLIPS, RM ;

SHARMA, SK .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1994, 4 (19) :2313-2316

[2]

AONO T, Patent No. 341104

[3]

ARISTOFF PA, 1990, Patent No. 9008143

[4]

Armand J, 1988, Prog Clin Biol Res, V280, P235

[5]

ATASSI G, 1985, EUR J MED CHEM, V20, P393

[6] POTENTIAL ANTITUMOR AGENTS .60. RELATIONSHIPS BETWEEN STRUCTURE AND INVIVO COLON 38 ACTIVITY FOR 5-SUBSTITUTED 9-OXOXANTHENE-4-ACETIC ACIDS [J].

ATWELL, GJ ;

REWCASTLE, GW ;

BAGULEY, BC ;

DENNY, WA .

JOURNAL OF MEDICINAL CHEMISTRY, 1990, 33 (05) :1375-1379

[7]

ATWELL GJ, 1989, ANTI-CANCER DRUG DES, V4, P161

[8] POTENTIAL ANTITUMOR AGENTS .57. 2-PHENYLQUINOLINE-8-CARBOXAMIDES AS MINIMAL DNA-INTERCALATING ANTITUMOR AGENTS WITH INVIVO SOLID TUMOR-ACTIVITY [J].

ATWELL, GJ ;

BAGULEY, BC ;

DENNY, WA .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (02) :396-401

[9] COMPARISON OF THE EFFECTS OF FLAVONE ACETIC-ACID, FOSTRIECIN, HOMOHARRINGTONINE AND TUMOR NECROSIS FACTOR-ALPHA ON COLON-38 TUMORS IN MICE [J].

BAGULEY, BC ;

CALVELEY, SB ;

CROWE, KK ;

FRAY, LM ;

OROURKE, SA ;

SMITH, GP .

EUROPEAN JOURNAL OF CANCER & CLINICAL ONCOLOGY, 1989, 25 (02) :263-269

[10]

Bibby M C, 1988, Prog Clin Biol Res, V280, P243

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