SYNTHESIS OF 16-ALPHA-[I-125]IODO-5-ALPHA-DIHYDROTESTOSTERONE AND EVALUATION OF ITS AFFINITY FOR THE ANDROGEN RECEPTOR

被引：25

作者：

HOYTE, RM

ROSNER, W

HOCHBERG, RB

机构：

[1] YALE UNIV,SCH MED,DEPT OBSTET & GYNECOL,REPROD BIOL SECT,NEW HAVEN,CT 06510

[2] YALE UNIV,SCH MED,DEPT MOLEC BIOL & BIOCHEM,NEW HAVEN,CT 06510

[3] COLUMBIA UNIV,ROOSEVELT HOSP,COLL PHYS & SURG,DEPT MED,NEW YORK,NY 10019

来源：

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY | 1982年 / 16卷 / 05期

关键词：

D O I：

10.1016/0022-4731(82)90097-8

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：621 / 628

页数：8

共 29 条

[1] CONFORMATION OF NON-AROMATIC RING COMPOUNDS .25. GEOMETRY AND CONFORMATION OF RING D IN SOME STEROIDS FROM X-RAY STRUCTURE DETERMINATIONS [J].

ALTONA, C ;

GEISE, HJ ;

ROMERS, C .

TETRAHEDRON, 1968, 24 (01) :13-&

[2]

ALTONA C, 1971, CONFORMATIONAL ANALY, P1

[3]

BROWN CA, 1974, J ORG CHEM, V39, P1324, DOI 10.1021/jo00923a042

[4] STEROID RING D TORSIONAL ANGLES AND CONFORMATIONS FROM X-RAY DATA [J].

BRUTCHER, FV ;

LEOPOLD, EJ .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1966, 88 (13) :3156-&

[5] SOME HYPOTHESESE ABOUT INTERACTIONS BETWEEN ESTROGEN AND ANDROGEN AND THEIR POSSIBLE RECEPTORS [J].

BUSETTA, B ;

COURSEILLE, C ;

PRECIGOUX, G ;

HOSPITAL, M .

JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1977, 8 (01) :63-67

[6]

COUNSELL RE, 1981, RADIOPHARMACEUTICALS, P425

[7] SPECTRA + STEREOCHEMISTRY .9. NUCLEAR MAGNETIC RESONANCE SPECTRAL STUDY OF SOME 16-SUBSTITUTED PREGNENES + 17 ALPHA-PREGNENES [J].

CROSS, AD ;

CRABBE, P .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1964, 86 (06) :1221-&

[8] STEROIDS .269. SPECTRA + STEREOCHEMISTRY .17. NONADDITIVITY OF ANGULAR METHYL PROTON FREQUENCY SHIFTS + RING D CONFORMATIONAL CHANGES IN 16-METHYL STEROIDS [J].

CROSS, AD ;

BEARD, C .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1964, 86 (23) :5317-&

[9] SYNTHESIS OF BR-77-LABELED 5ALPHA-DIHYDROTESTOSTERONE AND A COMPARISON OF ITS DISTRIBUTION IN RATS WITH BR-77-BROMIDE [J].

EAKINS, MN ;

WATERS, SL .

INTERNATIONAL JOURNAL OF APPLIED RADIATION AND ISOTOPES, 1979, 30 (11) :701-703

[10] CONFIGURATION OF STEROID BROMOKETONES .1. METHYL 4-BETA-BROMO-3-KETOCHOLANATE [J].

FIESER, LF ;

ETTORRE, R .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1953, 75 (07) :1700-1704

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