STRUCTURE-ACTIVITY RELATIONSHIP OF HISTAMINE ANALOGS .18. ABSOLUTE-CONFIGURATION AND HISTAMINE-LIKE ACTIVITY OF THE ENANTIOMERS OF 5-AMINO-4,5,6,7-TETRAHYDROBENZIMIDAZOLE

被引：9

作者：

SCHWARZ, S

SCHUNACK, W

机构：

[1] Fachbereich Pharmazie, Johannes Gutenberg-Universität, Mainz, 6500

来源：

ARCHIV DER PHARMAZIE | 1979年 / 312卷 / 11期

关键词：

D O I：

10.1002/ardp.19793121108

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

Es werden die Racemattrennung von 5‐Amino‐4,5,6,7‐tetrahydro‐benzimidazol 3, die Bestimmung der absoluten Konfiguration sowie die histaminartige Wirksamkeit der Enantiomere am Ileum (H1) und Atrium (H2) des Meerschweinchens beschrieben. Copyright © 1979 WILEY‐VCH Verlag GmbH & Co. KGaA, Weinheim

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页码：933 / 939

页数：7

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