ENDOGENOUS LIGANDS AND INVERSE AGONISM

被引：13

作者：

BAXTER, GS

TILFORD, NS

机构：

来源：

TRENDS IN PHARMACOLOGICAL SCIENCES | 1995年 / 16卷 / 08期

关键词：

D O I：

10.1016/S0165-6147(00)89038-0

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

页码：258 / 259

页数：2

共 7 条

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MILANO, CA ;

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APPARSUNDARAM, S ;

HYEK, MF ;

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[3]

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[4] ANTAGONISTS WITH NEGATIVE INTRINSIC ACTIVITY AT DELTA-OPIOID RECEPTORS COUPLED TO GTP-BINDING PROTEINS [J].

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[5] ESTIMATION OF PARTIAL AGONIST AFFINITY BY INTERACTION WITH A FULL AGONIST - A DIRECT OPERATIONAL MODEL-FITTING APPROACH [J].

LEFF, P ;

DOUGALL, IG ;

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[6] INVERSE AGONISM - PHARMACOLOGICAL CURIOSITY OR POTENTIAL THERAPEUTIC STRATEGY [J].

MILLIGAN, G ;

BOND, RA ;

LEE, M .

TRENDS IN PHARMACOLOGICAL SCIENCES, 1995, 16 (01) :10-13

[7]

SAMAMA P, 1994, MOL PHARMACOL, V45, P390

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