SYNTHESIS OF ACTIVATED 3-ARYLINDOLES

被引：47

作者：

BLACK, DS

BOWYER, MC

BOWYER, PK

IVORY, AJ

KIM, M

KUMAR, N

MCCONNELL, DB

POPIOLEK, M

机构：

来源：

AUSTRALIAN JOURNAL OF CHEMISTRY | 1994年 / 47卷 / 09期

关键词：

D O I：

10.1071/CH9941741

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A wide range of substituted 3-aryl-4,6-dimethoxyindoles (6) has been synthesized from the related alpha-anilinoacetophenones (5), in which the nitrogen atom is protected by a trifluoroacetyl or acetyl group. This method has led to the synthesis of a 3,7'-biindolyl (12).

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页码：1741 / 1750

页数：10

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