ASPARTYL ALPHA-((DIPHENYLPHOSPHINYL)OXY)METHYL KETONES AS NOVEL INHIBITORS OF INTERLEUKIN-1-BETA CONVERTING-ENZYME - UTILITY OF THE DIPHENYLPHOSPHINIC ACID LEAVING GROUP FOR THE INHIBITION OF CYSTEINE PROTEASES

被引:34
作者
DOLLE, RE [1 ]
SINGH, J [1 ]
WHIPPLE, D [1 ]
OSIFO, IK [1 ]
SPEIER, G [1 ]
GRAYBILL, TL [1 ]
GREGORY, JS [1 ]
HARRIS, AL [1 ]
HELASZEK, CT [1 ]
MILLER, RE [1 ]
ATOR, MA [1 ]
机构
[1] STERLING WINTHROP PHARMACEUT, DEPT BIOCHEM, DIV RES, COLLEGEVILLE, PA 19426 USA
关键词
D O I
10.1021/jm00002a002
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:220 / 222
页数:3
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