TRITIATED-6-BETA-FLUORO-6-DESOXY-OXYMORPHONE ([H-3] FOXY) - A NEW LIGAND AND PHOTOAFFINITY PROBE FOR THE MU OPIOID RECEPTORS

被引：16

作者：

ROTHMAN, RB

BYKOV, V

RICE, KC

JACOBSON, AE

KOOPER, GN

BOWEN, WD

机构：

[1] ST ELIZABETHS HOSP, NIMH, PRECLIN PHARMACOL LAB, WASHINGTON, DC 20032 USA

[2] NIDDK, NEUROSCI LAB, BETHESDA, MD 20892 USA

[3] BROWN UNIV, DIV BIOL & MED, BIOCHEM SECT, PROVIDENCE, RI 02912 USA

来源：

NEUROPEPTIDES | 1988年 / 11卷 / 01期

关键词：

D O I：

10.1016/0143-4179(88)90020-0

中图分类号：

R5 [内科学];

学科分类号：

1002 ; 100201 ;

摘要：

引用

页码：1 / 6

页数：6

共 26 条

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LOWRY OH, 1951, J BIOL CHEM, V193, P265

[9] POTENTIAL AFFINITY LABELS FOR THE OPIATE RECEPTOR BASED ON FENTANYL AND RELATED-COMPOUNDS [J].

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JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (08) :913-919

[10] HIGH AND LOW AFFINITY OPIOID BINDING-SITES - RELATIONSHIP TO MU-SITES AND DELTA-SITES [J].

PASTERNAK, GW .

LIFE SCIENCES, 1982, 31 (12-1) :1303-1306

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