A FACILE ONE-POT SYNTHESIS OF 5-TRIFLUOROMETHYLOXAZOLES AND 5-PERFLUOROALKYLOXAZOLES FROM N-ALKYL-N-ACYLAMINO ACIDS

被引：9

作者：

KAWASE, M

机构：

[1] Faculty of Pharmaceutical Sciences, Josai University, Sakado-shi, Saitama, 350-02

来源：

HETEROCYCLES | 1993年 / 36卷 / 11期

关键词：

D O I：

10.3987/COM-93-6508

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The reaction of N-acyl-N-benzyl-alpha-amino acids with trifluoroacetic or perfluorocarboxylic anhydride in the presence of pyridine affords 5-trifluoromethyl- or 5-perfluoroalkyloxazoles in high yields.

引用

页码：2441 / 2444

页数：4

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