PHOSPHORYLATION OF MU-OPIOID RECEPTORS - A PUTATIVE MECHANISM OF SELECTIVE UNCOUPLING OF RECEPTOR-GI INTERACTION, MEASURED WITH LOW-KM GTPASE AND NUCLEOTIDE-SENSITIVE AGONIST BINDING

被引:41
作者
HARADA, H
UEDA, H
WADA, Y
KATADA, T
UI, M
SATOH, M
机构
[1] KYOTO UNIV,FAC PHARMACEUT SCI,DEPT PHARMACOL,KYOTO 606,JAPAN
[2] TOKYO INST TECHNOL,DEPT LIFE SCI,YOKOHAMA,KANAGAWA 227,JAPAN
[3] UNIV TOKYO,FAC PHARMACEUT SCI,DEPT PHYSIOL CHEM,TOKYO 113,JAPAN
关键词
D O I
10.1016/0304-3940(89)90688-5
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:221 / 226
页数:6
相关论文
共 19 条
[1]   PERTUSSIS TOXIN TREATMENT MODIFIES OPIATE ACTION IN THE RAT-BRAIN STRIATUM [J].
ABOOD, ME ;
LAW, PY ;
LOH, HH .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 127 (02) :477-483
[3]   CATECHOLAMINE-STIMULATED GTPASE ACTIVITY IN TURKEY ERYTHROCYTE-MEMBRANES [J].
CASSEL, D ;
SELINGER, Z .
BIOCHIMICA ET BIOPHYSICA ACTA, 1976, 452 (02) :538-551
[4]   G-PROTEINS - TRANSDUCERS OF RECEPTOR-GENERATED SIGNALS [J].
GILMAN, AG .
ANNUAL REVIEW OF BIOCHEMISTRY, 1987, 56 :615-649
[5]   PHOSPHORYLATION OF BRAIN MUSCARINIC RECEPTOR - EVIDENCE OF RECEPTOR REGULATION [J].
HO, AKS ;
LING, QL ;
DUFFIELD, R ;
LAM, PH ;
WANG, JH .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1987, 142 (03) :911-918
[6]  
KATADA T, 1986, J BIOL CHEM, V261, P8182
[7]   A NEW GTP-BINDING PROTEIN IN BRAIN-TISSUES SERVING AS THE SPECIFIC SUBSTRATE OF ISLET-ACTIVATING PROTEIN, PERTUSSIS TOXIN [J].
KATADA, T ;
OINUMA, M ;
KUSAKABE, K ;
UI, M .
FEBS LETTERS, 1987, 213 (02) :353-358
[8]  
KOSKI G, 1982, J BIOL CHEM, V257, P4035
[9]  
KUROSE H, 1983, J BIOL CHEM, V258, P4870
[10]  
KWATRA MM, 1986, J BIOL CHEM, V261, P2429