MORPHINE-6-GLUCURONIDE - RECEPTOR-BINDING PROFILE IN BOVINE CAUDATE-NUCLEUS

被引:21
作者
CHRISTENSEN, CB
REIFF, L
机构
[1] Department of Pharmacology, University of Copenhagen, Copenhagen, DK-2100, 20, Juliane Maries Vej
来源
PHARMACOLOGY & TOXICOLOGY | 1991年 / 68卷 / 02期
关键词
D O I
10.1111/j.1600-0773.1991.tb02056.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:151 / 153
页数:3
相关论文
共 10 条
[1]   MORPHINE-6-GLUCURONIDE - ANALGESIC EFFECTS AND RECEPTOR-BINDING PROFILE IN RATS [J].
ABBOTT, FV ;
PALMOUR, RM .
LIFE SCIENCES, 1988, 43 (21) :1685-1695
[2]   MORPHINE-6-GLUCURONIDE HAS HIGH-AFFINITY FOR THE OPIOID RECEPTOR [J].
CHRISTENSEN, CB ;
JORGENSEN, LN .
PHARMACOLOGY & TOXICOLOGY, 1987, 60 (01) :75-76
[3]  
GOLDSTEIN A, 1989, MOL PHARMACOL, V36, P265
[4]   ANALGESIC EFFICACY AND CSF PHARMACOKINETICS OF INTRATHECAL MORPHINE-6-GLUCURONIDE - COMPARISON WITH MORPHINE [J].
HANNA, MH ;
PEAT, SJ ;
WOODHAM, M ;
KNIBB, A ;
FUNG, C .
BRITISH JOURNAL OF ANAESTHESIA, 1990, 64 (05) :547-550
[5]  
LATHI RA, 1985, EUR J PHARMACOL, V109, P281
[6]   BIS-PENICILLAMINE ENKEPHALINS POSSESS HIGHLY IMPROVED SPECIFICITY TOWARD DELTA-OPIOID RECEPTORS [J].
MOSBERG, HI ;
HURST, R ;
HRUBY, VJ ;
GEE, K ;
YAMAMURA, HI ;
GALLIGAN, JJ ;
BURKS, TF .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (19) :5871-5874
[7]   ENHANCED BINDING OF MORPHINE AND NALORPHINE TO OPIOID DELTA RECEPTOR BY GLUCURONATE AND SULFATE CONJUGATIONS AT THE 6-POSITION [J].
OGURI, K ;
YAMADAMORI, I ;
SHIGEZANE, J ;
HIRANO, T ;
YOSHIMURA, H .
LIFE SCIENCES, 1987, 41 (12) :1457-1464
[8]   MORPHINE-6-GLUCURONIDE, A POTENT MU AGONIST [J].
PASTERNAK, GW ;
BODNAR, RJ ;
CLARK, JA ;
INTURRISI, CE .
LIFE SCIENCES, 1987, 41 (26) :2845-2849
[9]  
PAUL D, 1989, J PHARMACOL EXP THER, V251, P477
[10]   ANALGESIC EFFECT OF MORPHINE GLUCURONIDES [J].
SHIMOMURA, K ;
KAMATA, O ;
UEKI, S ;
IDA, S ;
OGURI, K ;
YOSHIMURA, H ;
TSUKAMOTO, H .
TOHOKU JOURNAL OF EXPERIMENTAL MEDICINE, 1971, 105 (01) :45-52