ANTI-RETROVIRUS ACTIVITY OF 3'-FLUORO-SUBSTITUTED AND 3'-AZIDO-SUBSTITUTED PYRIMIDINE 2',3'-DIDEOXYNUCLEOSIDE ANALOGS

被引：213

作者：

BALZARINI, J

BABA, M

PAUWELS, R

HERDEWIJN, P

DECLERCO, E

机构：

来源：

BIOCHEMICAL PHARMACOLOGY | 1988年 / 37卷 / 14期

关键词：

D O I：

10.1016/0006-2952(88)90049-4

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

引用

收藏

页码：2847 / 2856

页数：10

相关论文

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[1] BOTH 2',3'-DIDEOXYTHYMIDINE AND ITS 2',3'-UNSATURATED DERIVATIVE (2',3'-DI-DEOXYTHYMIDINENE) ARE POTENT AND SELECTIVE INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS-REPLICATION INVITRO
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[2] THE INVITRO AND INVIVO ANTI-RETROVIRUS ACTIVITY, AND INTRACELLULAR METABOLISM OF 3'-AZIDO-2',3'-DIDEOXYTHYMIDINE AND 2',3'-DIDEOXYCYTIDINE ARE HIGHLY DEPENDENT ON THE CELL SPECIES
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[3] STRATEGIES FOR THE MEASUREMENT OF THE INHIBITORY EFFECTS OF THYMIDINE ANALOGS ON THE ACTIVITY OF THYMIDYLATE SYNTHASE IN INTACT MURINE LEUKEMIA L1210-CELLS
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[4] ROLE OF THYMIDINE KINASE IN THE INHIBITORY ACTIVITY OF 5-SUBSTITUTED-2'-DEOXYURIDINES ON THE GROWTH OF HUMAN AND MURINE TUMOR-CELL LINES
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[5] 5-SUBSTITUTED 2'-DEOXYURIDINES - CORRELATION BETWEEN INHIBITION OF TUMOR-CELL GROWTH AND INHIBITION OF THYMIDINE KINASE AND THYMIDYLATE SYNTHETASE
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[7] BALZARINI J, 1983, MOL PHARMACOL, V23, P175
[8] BROAD-SPECTRUM ANTIRETROVIRAL ACTIVITY OF 2',3'-DIDEOXYNUCLEOSIDES
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