METOPROLOL OXIDATION BY RAT-LIVER MICROSOMES - INHIBITION BY DEBRISOQUINE AND OTHER DRUGS

被引:22
作者
LENNARD, MS
CREWE, HK
TUCKER, GT
WOODS, HF
机构
关键词
D O I
10.1016/0006-2952(86)90186-3
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:2757 / 2761
页数:5
相关论文
共 39 条
[1]   ANIMAL MODELING OF HUMAN POLYMORPHIC DRUG OXIDATION - THE METABOLISM OF DEBRISOQUINE AND PHENACETIN IN RAT INBRED STRAINS [J].
ALDABBAGH, SG ;
IDLE, JR ;
SMITH, RL .
JOURNAL OF PHARMACY AND PHARMACOLOGY, 1981, 33 (03) :161-164
[2]   METABOLISM OF METOPROLOL IN RAT INVITRO AND INVIVO [J].
ARFWIDSSON, A ;
BORG, KO ;
HOFFMANN, KJ ;
SKANBERG, I .
XENOBIOTICA, 1976, 6 (11) :691-711
[3]   MONO-OXYGENASE ACTIVITY OF HUMAN-LIVER IN MICROSOMAL FRACTIONS OF NEEDLE-BIOPSY SPECIMENS [J].
BOOBIS, AR ;
BRODIE, MJ ;
KAHN, GC ;
FLETCHER, DR ;
SAUNDERS, JH ;
DAVIES, DS .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 9 (01) :11-19
[4]  
BOOBIS AR, 1983, MOL PHARMACOL, V23, P474
[5]   GENETIC-POLYMORPHISM IN DRUG OXIDATION - INVITRO STUDIES OF HUMAN DEBRISOQUINE 4-HYDROXYLASE AND BUFURALOL 1'-HYDROXYLASE ACTIVITIES [J].
BOOBIS, AR ;
MURRAY, S ;
HAMPDEN, CE ;
DAVIES, DS .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (01) :65-71
[6]  
BORG KO, 1975, ACTA PHARMACOL TOX, V36, P125
[7]  
Cornish-Bowden A., 1979, FUNDAMENTALS ENZYME
[8]   EVIDENCE FOR AN ENZYMATIC DEFECT IN THE 4-HYDROXYLATION OF DEBRISOQUINE BY HUMAN-LIVER [J].
DAVIES, DS ;
KAHN, GC ;
MURRAY, S ;
BRODIE, MJ ;
BOOBIS, AR .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1981, 11 (01) :89-91
[9]   DEFECTIVE HYDROXYLATION OF BUFURALOL ASSOCIATED WITH SIDE-EFFECTS OF THE DRUG IN POOR METABOLIZERS [J].
DAYER, P ;
KUBLI, A ;
KUPFER, A ;
COURVOISIER, F ;
BALANT, L ;
FABRE, J .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1982, 13 (05) :750-752
[10]   CHARACTERIZATION OF A HUMAN-LIVER CYTOCHROME-P-450 INVOLVED IN THE OXIDATION OF DEBRISOQUINE AND OTHER DRUGS BY USING ANTIBODIES RAISED TO THE ANALOGOUS RAT ENZYME [J].
DISTLERATH, LM ;
GUENGERICH, FP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1984, 81 (23) :7348-7352