ANTICONVULSANT ACTIVITY OF THE GLIAL GABA UPTAKE INHIBITOR, THAO, IN CHEMICAL SEIZURES

被引:16
作者
GONSALVES, SF
TWITCHELL, B
HARBAUGH, RE
KROGSGAARDLARSEN, P
SCHOUSBOE, A
机构
[1] UNIV COPENHAGEN,PANUM INST,DEPT BIOCHEM A,PHARMABIOTEC RES CTR,DK-2200 COPENHAGEN N,DENMARK
[2] DARTMOUTH COLL,HITCHCOCK MED CTR,DEPT SURG,HANOVER,NH 03756
[3] DARTMOUTH COLL,HITCHCOCK MED CTR,DEPT PHARMACOL,HANOVER,NH 03756
[4] ROYAL DANISH SCH PHARM,DEPT CHEM BC,PHARMABIOTEC RES CTR,DK-2100 COPENHAGEN,DENMARK
关键词
D O I
10.1016/0014-2999(89)90576-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:265 / 268
页数:4
相关论文
共 10 条
[1]   ANTI-CONVULSANT ACTIVITY OF GABA UPTAKE INHIBITORS AND THEIR PRODRUGS FOLLOWING CENTRAL OR SYSTEMIC ADMINISTRATION [J].
CROUCHER, MJ ;
MELDRUM, BS ;
KROGSGAARDLARSEN, P .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1983, 89 (3-4) :217-228
[2]  
GONSALVES SF, IN PRESS EPILEPSY RE, V3
[3]   CONVULSANT AND ANTICONVULSANT ACTIONS IN DBA-2 MICE OF COMPOUNDS BLOCKING THE REUPTAKE OF GABA [J].
HORTON, RW ;
COLLINS, JF ;
ANLEZARK, GM ;
MELDRUM, BS .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1979, 59 (1-2) :75-83
[4]   MUSCIMOL ANALOGS .2. SYNTHESIS OF SOME BICYCLIC 3-ISOXAZOLOL ZWITTERIONS [J].
KROGSGAARDLARSEN, P .
ACTA CHEMICA SCANDINAVICA SERIES B-ORGANIC CHEMISTRY AND BIOCHEMISTRY, 1977, 31 (07) :584-588
[5]   ON THE MEASUREMENT IN RATS OF THE CONVULSANT EFFECT OF DRUGS AND THE CHANGES WHICH FOLLOW ELECTROCONVULSIVE SHOCK [J].
NUTT, DJ ;
COWEN, PJ ;
GREEN, AR .
NEUROPHARMACOLOGY, 1980, 19 (10) :1017-1023
[6]  
SCHOUSBOE A, 1986, J NEUROCHEM, V47, P758
[7]   TRANSPORT AND METABOLISM OF GAMMA AMINOBUTYRIC-ACID IN NEURONS AND GLIA - IMPLICATIONS FOR EPILEPSY [J].
SCHOUSBOE, A ;
LARSSON, OM ;
WOOD, JD ;
KROGSGAARDLARSEN, P .
EPILEPSIA, 1983, 24 (05) :531-538
[8]   HETEROCYCLIC GABA ANALOGS AS NEW SELECTIVE INHIBITORS OF ASTROGLIAL GABA TRANSPORT [J].
SCHOUSBOE, A ;
LARSSON, OM ;
HERTZ, L ;
KROGSGAARDLARSEN, P .
DRUG DEVELOPMENT RESEARCH, 1981, 1 (02) :115-127
[9]   INVIVO CHANGES IN THE GABA CONTENT OF NERVE-ENDINGS (SYNAPTOSOMES) INDUCED BY INHIBITORS OF GABA UPTAKE [J].
WOOD, JD ;
SCHOUSBOE, A ;
KROGSGAARDLARSEN, P .
NEUROPHARMACOLOGY, 1980, 19 (11) :1149-1152
[10]  
YUNGER LM, 1984, J PHARMACOL EXP THER, V228, P109