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SELECTIVE AND ENANTIOSPECIFIC ACYLATION OF KAPPA-OPIOID RECEPTORS BY (1S,2S)-TRANS-2-ISOTHIOCYANATO-N-METHYL-N-[2-(1-PYRROLIDINYL)CYCLOHEXYL]BENZENEACETAMIDE - DEMONSTRATION OF KAPPA-RECEPTOR HETEROGENEITY
被引:40
作者
:
DECOSTA, BR
论文数:
0
引用数:
0
h-index:
0
机构:
NIDDKD,NEUROSCI LAB,DRUG DESIGN & SYNTH SECT,BETHESDA,MD 20892
DECOSTA, BR
ROTHMAN, RB
论文数:
0
引用数:
0
h-index:
0
机构:
NIDDKD,NEUROSCI LAB,DRUG DESIGN & SYNTH SECT,BETHESDA,MD 20892
ROTHMAN, RB
BYKOV, V
论文数:
0
引用数:
0
h-index:
0
机构:
NIDDKD,NEUROSCI LAB,DRUG DESIGN & SYNTH SECT,BETHESDA,MD 20892
BYKOV, V
JACOBSON, AE
论文数:
0
引用数:
0
h-index:
0
机构:
NIDDKD,NEUROSCI LAB,DRUG DESIGN & SYNTH SECT,BETHESDA,MD 20892
JACOBSON, AE
RICE, KC
论文数:
0
引用数:
0
h-index:
0
机构:
NIDDKD,NEUROSCI LAB,DRUG DESIGN & SYNTH SECT,BETHESDA,MD 20892
RICE, KC
机构
:
[1]
NIDDKD,NEUROSCI LAB,DRUG DESIGN & SYNTH SECT,BETHESDA,MD 20892
[2]
NIMH,CLIN STUDIES LAB,RECEPTOR STUDIES UNIT,BETHESDA,MD 20892
来源
:
JOURNAL OF MEDICINAL CHEMISTRY
|
1989年
/ 32卷
/ 02期
关键词
:
D O I
:
10.1021/jm00122a001
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:281 / 283
页数:3
相关论文
共 30 条
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PORTOGHESE, PS
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引用数:
0
h-index:
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机构:
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
PORTOGHESE, PS
LARSON, DL
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h-index:
0
机构:
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
LARSON, DL
JIANG, JB
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
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PORTOGHESE, PS
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
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LARSON, DL
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TAKEMORI, AE
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
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PORTOGHESE, PS
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
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6-BETA [N,N-BIS(2-CHLOROETHYL)AMINO]-17-(CYCLOPROPYLMETHYL)-4,5-ALPHA-EPOXY-3,14-DIHYDROXYMORPHINAN (CHLORANALTREXAMINE) - POTENT OPIOID RECEPTOR ALKYLATING AGENT WITH ULTRALONG NARCOTIC-ANTAGONIST ACTIVITY
PORTOGHESE, PS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
PORTOGHESE, PS
LARSON, DL
论文数:
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引用数:
0
h-index:
0
机构:
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
LARSON, DL
JIANG, JB
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
TAKEMORI, AE
CARUSO, TP
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0
h-index:
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
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PORTOGHESE, PS
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引用数:
0
h-index:
0
机构:
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
PORTOGHESE, PS
LARSON, DL
论文数:
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引用数:
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h-index:
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机构:
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
LARSON, DL
SAYRE, LM
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h-index:
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
SAYRE, LM
FRIES, DS
论文数:
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
FRIES, DS
TAKEMORI, AE
论文数:
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引用数:
0
h-index:
0
机构:
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
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PORTOGHESE, PS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
PORTOGHESE, PS
NAGASE, H
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
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UNIV MINNESOTA,SCH MED,DEPT PHARMACOL,MINNEAPOLIS,MN 55455
LIPKOWSKI, AW
LARSON, DL
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0
引用数:
0
h-index:
0
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