A STEREOSELECTIVE SYNTHESIS OF A NOVEL MODEL-COMPOUND OF CARZINOPHILIN CARRYING THE C6-C-13 UNIT WITH CORRECT STEREOCHEMISTRY

被引：26

作者：

HASHIMOTO, M ^{[1
]}

TERASHIMA, S ^{[1
]}

机构：

[1] SAGAMI CHEM RES CTR, SAGAMIHARA, KANAGAWA 229, JAPAN

来源：

CHEMISTRY LETTERS | 1994年 / 06期

关键词：

D O I：

10.1246/cl.1994.1001

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The title synthesis was achieved by featuring stereocontrolled elaboration of the functionalized pyrrolidine-2-thione from 2,3,5-tri-O-benzyl-beta-D-arabinofuranose and base-induced construction of an aziridine ring from the 5-mesyloxymethylpyrrolidine.

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页码：1001 / 1002

页数：2

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