SYNTHESIS AND BIOLOGICAL-ACTIVITIES OF CONDENSED HETEROCYCLO[N,M-A,B, OR C]QUINAZOLINES

被引:37
作者
SHABAN, MAE [1 ]
TAHA, MAM [1 ]
SHARSHIRA, EM [1 ]
机构
[1] UNIV ALEXANDRIA,FAC SCI,DEPT CHEM,ALEXANDRIA,EGYPT
关键词
D O I
10.1016/S0065-2725(08)60963-0
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The synthesis and biological activities of title compounds are systematically arranged according to the complexity of the heterocyclic ring directly fused to the pyrimidine ring of the quinazoline nucleus (irrespective of other rings that might be fused to it), starting with those having one nitrogen atom in a three-membered ring and going to more complex ones. The heterocycles have been arranged according to the type of their heteroatom in the following order: nitrogen, oxygen, sulfur, and selenium. Consideration has been given to the alternative nomenclature of some heterocyclo- quinazolines, also known as quinazolinoheterocycles, in order to comply with the nomenclature rules of the IUPAC. The diverse biological activities of the title compounds have certainly contributed to the extensive efforts directed towards their synthesis. © 1991 Academic Press Inc.
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页码:1 / 153
页数:153
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