ACTIVATION OF BRAIN-FUNCTION BY S-135, A BENZODIAZEPINE RECEPTOR INVERSE AGONIST

被引:14
作者
MATSUSHITA, A [1 ]
KAWASAKI, K [1 ]
MATSUBARA, K [1 ]
EIGYO, M [1 ]
SHINDO, H [1 ]
TAKADA, S [1 ]
机构
[1] SHIONOGI & CO LTD,SHIONOGI RES LAB,DIV CHEM,FUKUSHIMA KU,OSAKA 553,JAPAN
关键词
D O I
10.1016/0278-5846(88)90091-7
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:951 / 966
页数:16
相关论文
共 31 条
[21]  
LITTLE H J, 1986, British Journal of Pharmacology, V89, p800P
[22]  
MATSUSHITA A, 1987, J PHARMACOBIO-DYNAM, V10, pS165
[23]  
MATSUSHITA A, 1986, 15TH P CINP C SAN JU, P42
[24]  
Pellegrino LJ., 1967, STEREOTAXIC ATLAS RA
[25]   PROCONFLICT EFFECT OF BENZODIAZEPINE RECEPTOR INVERSE AGONISTS AND OTHER INHIBITORS OF GABA FUNCTION [J].
PETERSEN, EN ;
JENSEN, LH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 103 (1-2) :91-97
[26]   DEPRESSION - NEW ANIMAL-MODEL SENSITIVE TO ANTIDEPRESSANT TREATMENTS [J].
PORSOLT, RD ;
LEPICHON, M ;
JALFRE, M .
NATURE, 1977, 266 (5604) :730-732
[27]   [DEOXYGLUCOSE-C-14 METHOD FOR MEASUREMENT OF LOCAL CEREBRAL GLUCOSE-UTILIZATION - THEORY, PROCEDURE, AND NORMAL VALUES IN CONSCIOUS AND ANESTHETIZED ALBINO-RAT [J].
SOKOLOFF, L ;
REIVICH, M ;
KENNEDY, C ;
DESROSIERS, MH ;
PATLAK, CS ;
PETTIGREW, KD ;
SAKURADA, O ;
SHINOHARA, M .
JOURNAL OF NEUROCHEMISTRY, 1977, 28 (05) :897-916
[28]   A NEW THIENYLPYRAZOLOQUINOLINE - A POTENT AND ORALLY ACTIVE INVERSE AGONIST TO BENZODIAZEPINE RECEPTORS [J].
TAKADA, S ;
SHINDO, H ;
SASATANI, T ;
MATSUSHITA, A ;
EIGYO, M ;
KAWASAKI, K ;
MURATA, S .
JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (03) :454-455
[29]  
TENNEN S, 1980, NATURE, V288, P609
[30]   BENZODIAZEPINE IMPAIRS AND BETA-CARBOLINE ENHANCES PERFORMANCE IN LEARNING AND MEMORY TASKS [J].
VENAULT, P ;
CHAPOUTHIER, G ;
DECARVALHO, LP ;
SIMIAND, J ;
MORRE, M ;
DODD, RH ;
ROSSIER, J .
NATURE, 1986, 321 (6073) :864-866