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TARGETS AND STRATEGIES FOR THE ANTIVIRAL CHEMOTHERAPY OF AIDS
被引:103
作者
:
DECLERCQ, E
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT MICROBIOL,B-3000 LOUVAIN,BELGIUM
DECLERCQ, E
机构
:
[1]
DEPT MICROBIOL,B-3000 LOUVAIN,BELGIUM
[2]
REGA INST,B-3000 LOUVAIN,BELGIUM
来源
:
TRENDS IN PHARMACOLOGICAL SCIENCES
|
1990年
/ 11卷
/ 05期
关键词
:
D O I
:
10.1016/0165-6147(90)90115-O
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
Eradication of human immunodeficiency virus (HIV) from infected cells or organisms has remained an elusive goal. In principle, any of the steps in the replicative cycle could form the basis for rational design of chemotherapeutic agents, although in practice not all have so far proved amenable to intervention. Here, Erik De Clercq summarizes the strategies that are being employed, focusing primarily on recent promising developments in inhibition of adsorption of HIV onto CD4+ T cells, and inhibition of the viral reverse transcriptase. © 1990.
引用
收藏
页码:198 / 205
页数:8
相关论文
共 37 条
[31]
ANTIVIRAL AGENTS TARGETED TO INTERACT WITH VIRAL CAPSID PROTEINS AND A POSSIBLE APPLICATION TO HUMAN IMMUNODEFICIENCY VIRUS
ROSSMANN, MG
论文数:
0
引用数:
0
h-index:
0
ROSSMANN, MG
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1988,
85
(13)
: 4625
-
4627
[32]
SYNCYTIUM FORMATION AND DESTRUCTION OF BYSTANDER CD4+ CELLS COCULTURED WITH T-CELLS PERSISTENTLY INFECTED WITH HUMAN IMMUNODEFICIENCY VIRUS AS DEMONSTRATED BY FLOW-CYTOMETRY
SCHOLS, D
论文数:
0
引用数:
0
h-index:
0
SCHOLS, D
PAUWELS, R
论文数:
0
引用数:
0
h-index:
0
PAUWELS, R
BABA, M
论文数:
0
引用数:
0
h-index:
0
BABA, M
DESMYTER, J
论文数:
0
引用数:
0
h-index:
0
DESMYTER, J
DECLERCQ, E
论文数:
0
引用数:
0
h-index:
0
DECLERCQ, E
[J].
JOURNAL OF GENERAL VIROLOGY,
1989,
70
: 2397
-
2408
[33]
SCHOLS D, 1989, J ACQ IMMUN DEF SYND, V2, P10
[34]
SPECIFIC INTERACTION OF AURINTRICARBOXYLIC ACID WITH THE HUMAN IMMUNODEFICIENCY VIRUS CD4 CELL-RECEPTOR
SCHOLS, D
论文数:
0
引用数:
0
h-index:
0
SCHOLS, D
BABA, M
论文数:
0
引用数:
0
h-index:
0
BABA, M
PAUWELS, R
论文数:
0
引用数:
0
h-index:
0
PAUWELS, R
DESMYTER, J
论文数:
0
引用数:
0
h-index:
0
DESMYTER, J
DECLERCQ, E
论文数:
0
引用数:
0
h-index:
0
DECLERCQ, E
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1989,
86
(09)
: 3322
-
3326
[35]
SCHOLS D, IN PRESS VIROLOGY
[36]
ROLE OF THE HTLV-III/LAV ENVELOPE IN SYNCYTIUM FORMATION AND CYTOPATHICITY
SODROSKI, J
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
SODROSKI, J
GOH, WC
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
GOH, WC
ROSEN, C
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
ROSEN, C
CAMPBELL, K
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
CAMPBELL, K
HASELTINE, WA
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HASELTINE, WA
[J].
NATURE,
1986,
322
(6078)
: 470
-
474
[37]
3'-AZIDO-3'-DEOXYTHYMIDINE TRIPHOSPHATE AS AN INHIBITOR AND SUBSTRATE OF PURIFIED HUMAN-IMMUNODEFICIENCY-VIRUS REVERSE-TRANSCRIPTASE
STCLAIR, MH
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
STCLAIR, MH
RICHARDS, CA
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
RICHARDS, CA
SPECTOR, T
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
SPECTOR, T
WEINHOLD, KJ
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
WEINHOLD, KJ
MILLER, WH
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
MILLER, WH
LANGLOIS, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
LANGLOIS, AJ
FURMAN, PA
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
FURMAN, PA
[J].
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY,
1987,
31
(12)
: 1972
-
1977
←
1
2
3
4
→
共 37 条
[31]
ANTIVIRAL AGENTS TARGETED TO INTERACT WITH VIRAL CAPSID PROTEINS AND A POSSIBLE APPLICATION TO HUMAN IMMUNODEFICIENCY VIRUS
ROSSMANN, MG
论文数:
0
引用数:
0
h-index:
0
ROSSMANN, MG
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1988,
85
(13)
: 4625
-
4627
[32]
SYNCYTIUM FORMATION AND DESTRUCTION OF BYSTANDER CD4+ CELLS COCULTURED WITH T-CELLS PERSISTENTLY INFECTED WITH HUMAN IMMUNODEFICIENCY VIRUS AS DEMONSTRATED BY FLOW-CYTOMETRY
SCHOLS, D
论文数:
0
引用数:
0
h-index:
0
SCHOLS, D
PAUWELS, R
论文数:
0
引用数:
0
h-index:
0
PAUWELS, R
BABA, M
论文数:
0
引用数:
0
h-index:
0
BABA, M
DESMYTER, J
论文数:
0
引用数:
0
h-index:
0
DESMYTER, J
DECLERCQ, E
论文数:
0
引用数:
0
h-index:
0
DECLERCQ, E
[J].
JOURNAL OF GENERAL VIROLOGY,
1989,
70
: 2397
-
2408
[33]
SCHOLS D, 1989, J ACQ IMMUN DEF SYND, V2, P10
[34]
SPECIFIC INTERACTION OF AURINTRICARBOXYLIC ACID WITH THE HUMAN IMMUNODEFICIENCY VIRUS CD4 CELL-RECEPTOR
SCHOLS, D
论文数:
0
引用数:
0
h-index:
0
SCHOLS, D
BABA, M
论文数:
0
引用数:
0
h-index:
0
BABA, M
PAUWELS, R
论文数:
0
引用数:
0
h-index:
0
PAUWELS, R
DESMYTER, J
论文数:
0
引用数:
0
h-index:
0
DESMYTER, J
DECLERCQ, E
论文数:
0
引用数:
0
h-index:
0
DECLERCQ, E
[J].
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1989,
86
(09)
: 3322
-
3326
[35]
SCHOLS D, IN PRESS VIROLOGY
[36]
ROLE OF THE HTLV-III/LAV ENVELOPE IN SYNCYTIUM FORMATION AND CYTOPATHICITY
SODROSKI, J
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
SODROSKI, J
GOH, WC
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
GOH, WC
ROSEN, C
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
ROSEN, C
CAMPBELL, K
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
CAMPBELL, K
HASELTINE, WA
论文数:
0
引用数:
0
h-index:
0
机构:
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HARVARD UNIV,SCH PUBL HLTH,DEPT CANC BIOL,BOSTON,MA 02115
HASELTINE, WA
[J].
NATURE,
1986,
322
(6078)
: 470
-
474
[37]
3'-AZIDO-3'-DEOXYTHYMIDINE TRIPHOSPHATE AS AN INHIBITOR AND SUBSTRATE OF PURIFIED HUMAN-IMMUNODEFICIENCY-VIRUS REVERSE-TRANSCRIPTASE
STCLAIR, MH
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
STCLAIR, MH
RICHARDS, CA
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
RICHARDS, CA
SPECTOR, T
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
SPECTOR, T
WEINHOLD, KJ
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
WEINHOLD, KJ
MILLER, WH
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
MILLER, WH
LANGLOIS, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
LANGLOIS, AJ
FURMAN, PA
论文数:
0
引用数:
0
h-index:
0
机构:
BURROUGHS WELLCOME CO,DEPT MICROBIOL,RES TRIANGLE PK,NC 27709
FURMAN, PA
[J].
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY,
1987,
31
(12)
: 1972
-
1977
←
1
2
3
4
→