DESIGN AND SYNTHESIS OF A PROTOTYPICAL NONPEPTIDIC INHIBITOR MODEL FOR THE ENZYME RENIN

被引:31
作者
HANESSIAN, S
RAGHAVAN, S
机构
[1] Department of Chemistry, Montréal, Que. H3C 3J7, Universite Montreal P.O. Box 6128, Succ. Centre-ville
关键词
D O I
10.1016/S0960-894X(00)80364-9
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
The synthesis of non-peptidic acyclic and conformationally constrained compounds is described with the intention of designing models and chemical intermediates, for an inhibitor of the enzyme renin.
引用
收藏
页码:1697 / 1702
页数:6
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