Solid-phase synthesis of indoles using the palladium-catalysed coupling of alkynes with iodoaniline derivatives.

被引：119

作者：

Fagnola, MC ^{[1
]}

Candiani, I ^{[1
]}

Visentin, G ^{[1
]}

Cabri, W ^{[1
]}

Zarini, F ^{[1
]}

Mongelli, N ^{[1
]}

Bedeschi, A ^{[1
]}

机构：

[1] PHARMACIA & UPJOHN INC,ONCOL,I-20014 NERVIANO,MI,ITALY

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 13期

关键词：

D O I：

10.1016/S0040-4039(97)00300-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The solid-phase synthesis of indoles using Pd(0) catalysed coupling of alkynes with iodaniline derivatives is described. The reaction gives indoles in high yields with a wide range of alkynes. (C) 1997 Elsevier Science Ltd.

引用

页码：2307 / 2310

页数：4

共 18 条

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