Nonpeptide angiotensin II receptor antagonists: The next generation in antihypertensive therapy

被引:310
作者
Wexler, RR
Greenlee, WJ
Irvin, JD
Goldberg, MR
Prendergast, K
Smith, RD
Timmermans, PBMWM
机构
[1] DUPONT MERCK PHARMACEUT CO, WILMINGTON, DE 19880 USA
[2] MERCK SHARP & DOHME RES LABS, BLUE BELL, PA USA
[3] MERCK & CO INC, MERCK SHARP & DOHME RES LABS, RAHWAY, NJ 07065 USA
关键词
D O I
10.1021/jm9504722
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:625 / 656
页数:32
相关论文
共 340 条
  • [51] DUP-532 - A 2ND GENERATION OF NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONISTS
    CHIU, AT
    CARINI, DJ
    DUNCIA, JV
    LEUNG, KH
    MCCALL, DE
    PRICE, WA
    WONG, PC
    SMITH, RD
    WEXLER, RR
    TIMMERMANS, PBMWM
    CHANG, RSL
    LOTTI, VJ
    [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1991, 177 (01) : 209 - 217
  • [52] CHIU AT, 1990, J PHARMACOL EXP THER, V252, P711
  • [53] IDENTIFICATION OF ANGIOTENSIN-II RECEPTOR SUBTYPES
    CHIU, AT
    HERBLIN, WF
    MCCALL, DE
    ARDECKY, RJ
    CARINI, DJ
    DUNCIA, JV
    PEASE, LJ
    WONG, PC
    WEXLER, RR
    JOHNSON, AL
    TIMMERMANS, PBMWM
    [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1989, 165 (01) : 196 - 203
  • [54] NON-PEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONISTS .2. PHARMACOLOGY OF S-8308
    CHIU, AT
    CARINI, DJ
    JOHNSON, AL
    MCCALL, DE
    PRICE, WA
    THOOLEN, MJMC
    WONG, PC
    TABER, RI
    TIMMERMANS, PBMWM
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 157 (01) : 13 - 21
  • [55] CHRIST DD, 1990, OCT INT SOC STUD XEN, P137
  • [56] ORAL-ADMINISTRATION OF DUP-753, A SPECIFIC ANGIOTENSIN-II RECEPTOR ANTAGONIST, TO NORMAL-MALE VOLUNTEERS - INHIBITION OF PRESSOR-RESPONSE TO EXOGENOUS ANGIOTENSIN-I AND ANGIOTENSIN-II
    CHRISTEN, Y
    WAEBER, B
    NUSSBERGER, J
    PORCHET, M
    BORLAND, RM
    LEE, RJ
    MAGGON, K
    SHUM, L
    TIMMERMANS, PBMWM
    BRUNNER, HR
    [J]. CIRCULATION, 1991, 83 (04) : 1333 - 1342
  • [57] EFFECTS OF IRBESARTAN (SR 47436/BMS-186295) ON ANGIOTENSIN-II-INDUCED PRESSOR-RESPONSES IN THE PITHED RAT - POTENTIAL MECHANISMS OF ACTION
    CHRISTOPHE, B
    LIBON, R
    CAZAUBON, C
    NISATO, D
    MANNING, A
    CHATELAIN, P
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1995, 281 (02) : 161 - 171
  • [58] CLOAREC A, 1994, CAN J PHYSL PHARM S1, V72, P129
  • [59] COMPARISON OF ANGIOTENSIN-CONVERTING ENZYME-INHIBITION WITH ANGIOTENSIN-II RECEPTOR ANTAGONISM IN THE HUMAN FOREARM
    COCKCROFT, JR
    SCIBERRAS, DG
    GOLDBERG, MR
    RITTER, JM
    [J]. JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1993, 22 (04) : 579 - 584
  • [60] THE CLINICAL POTENTIAL OF RENIN INHIBITORS AND ANGIOTENSIN ANTAGONISTS
    CODY, RJ
    [J]. DRUGS, 1994, 47 (04) : 586 - 598