Comprehensive Survey of Chemical Libraries for Drug Discovery and Chemical Biology: 2007

被引:86
作者
Dolle, Roland E. [1 ]
Le Bourdonnec, Bertrand [1 ]
Goodman, Allan J. [1 ]
Morales, Guillermo A. [2 ]
Thomas, Craig J. [3 ]
Zhang, Wei [4 ]
机构
[1] Adolor Corp, Exton, PA 19341 USA
[2] Semafore Pharmaceut Inc, Indianapolis, IN 46268 USA
[3] NHGRI, NIH, Chem Genom Ctr, Rockville, MD 20850 USA
[4] Univ Massachusetts, Dept Chem, Boston, MA 02125 USA
来源
JOURNAL OF COMBINATORIAL CHEMISTRY | 2008年 / 10卷 / 06期
关键词
D O I
10.1021/cc800119z
中图分类号
O69 [应用化学];
学科分类号
081704 ;
摘要
[No abstract available]
引用
收藏
页码:753 / 802
页数:50
相关论文
共 530 条
[61]   Image-based chemical screening [J].
Carpenter, Anne E. .
NATURE CHEMICAL BIOLOGY, 2007, 3 (08) :461-465
[62]   Microwave-mediated heterocyclization to benzimidazo[2,1-b]quinazolin-12(5H)-ones [J].
Carpenter, Richard D. ;
Lam, Kit S. ;
Kurth, Mark J. .
JOURNAL OF ORGANIC CHEMISTRY, 2007, 72 (01) :284-287
[63]   Automated liquid-liquid extraction workstation for library synthesis and its use in the parallel and chromatography-free synthesis of 2-Alkyl-3-alkyl-4-(3H)-quinazolinones [J].
Carpintero, Mercedes ;
Cifuentes, Marta ;
Ferritto, Rafael ;
Haro, Ruben ;
Toledo, Miguel A. .
JOURNAL OF COMBINATORIAL CHEMISTRY, 2007, 9 (05) :818-822
[64]   Small-molecule inhibitors of protein geranylgeranyltransferase type I [J].
Castellano, Sabrina ;
Fiji, Hannah D. G. ;
Kinderman, Sape S. ;
Watanabe, Masaru ;
de Leon, Pablo ;
Tamanoi, Fuyuhiko ;
Kwon, Ohyun .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2007, 129 (18) :5843-+
[65]   Discovery of a series of 6,7-dimethoxy-4-pyrrolidylquinazoline PDE10A inhibitors [J].
Chappie, Thomas A. ;
Humphrey, John M. ;
Allen, Martin P. ;
Estep, Kimberly G. ;
Fox, Carol B. ;
Lebel, Lorraine A. ;
Liras, Spiros ;
Marr, Eric S. ;
Menniti, Frank S. ;
Pandit, Jayvardhan ;
Schmidt, Christopher J. ;
Tu, Meihua ;
Williams, Robert D. ;
Yang, Feng V. .
JOURNAL OF MEDICINAL CHEMISTRY, 2007, 50 (02) :182-185
[66]   Antiproliferative activities of a library of hybrids between indanones and HDAC inhibitor SAHA and MS-275 analogues [J].
Charrier, Cedric ;
Roche, Joeelle ;
Gesson, Jean-Pierre ;
Bertrand, Philippe .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 17 (22) :6142-6146
[67]   A versatile solid-phase synthesis of 3-aryl-1,2,4-oxadiazolones and analogues [J].
Charton, Julie ;
Cousaert, Nicolas ;
Bochu, Christophe ;
Willand, Nicolas ;
Deprez, Benoit ;
Deprez-Poulain, Rebecca .
TETRAHEDRON LETTERS, 2007, 48 (08) :1479-1483
[68]   One-step synthesis of oxazoline and dihydrooxazine libraries [J].
Chaudhry, Priyanka ;
Schoenen, Frank ;
Neuenswander, Benjamin ;
Lushington, Gerald H. ;
Aube, Jeffrey .
JOURNAL OF COMBINATORIAL CHEMISTRY, 2007, 9 (03) :473-476
[69]   One-pot synthesis of quinoline-based tetracycles by a tandem three-component reaction [J].
Che, Chao ;
Xiang, Jing ;
Wang, Guo-Xin ;
Fathi, Reza ;
Quan, Jun-Min ;
Yang, Zhen .
JOURNAL OF COMBINATORIAL CHEMISTRY, 2007, 9 (06) :982-989
[70]   Design of mutation-resistant HIV protease inhibitors with the substrate envelope hypothesis [J].
Chellappan, Sripriya ;
Reddy, G. S. Kiran Kumar ;
Ali, Akbar ;
Nalam, Madhavi N. L. ;
Anjum, Saima Ghafoor ;
Cao, Hong ;
Kairys, Visvaldas ;
Fernandes, Miguel X. ;
Altman, Michael D. ;
Tidor, Bruce ;
Rana, Tariq M. ;
Schiffer, Celia A. ;
Gilson, Michael K. .
CHEMICAL BIOLOGY & DRUG DESIGN, 2007, 69 (05) :298-313