First syntheses of C-4 methyl ether paclitaxel analogs and the unexpected reactivity of 4-deacetyl-4-methyl ether baccatin III

被引：8

作者：

Chen, SH ^{[1
]}

机构：

[1] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,WALLINGFORD,CT 06492

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 23期

关键词：

D O I：

10.1016/0040-4039(96)00746-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：3935 / 3938

页数：4

共 14 条

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[3]

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[4]

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[6]

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[7] SELECTIVE C-2 AND C-4 DEACYLATION AND ACYLATION OF TAXOL - THE FIRST SYNTHESIS OF A C-4 SUBSTITUTED TAXOL ANALOG [J].

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[8]

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[9] THE CHEMISTRY OF TAXOL, A CLINICALLY USEFUL ANTICANCER AGENT [J].

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[10] SYNTHESIS AND BIOLOGICAL EVALUATION OF 4-DEACETYLPACLITAXEL [J].

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GHARPURE, MM ;

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HAMEL, E .

TETRAHEDRON LETTERS, 1994, 35 (37) :6839-6842

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