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Selective androgen receptor modulators (SARMs): A novel approach to androgen therapy for the new millennium
被引:197
作者
:
Negro-Vilar, A
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, San Diego, CA 92121 USA
Ligand Pharmaceut Inc, San Diego, CA 92121 USA
Negro-Vilar, A
[
1
]
机构
:
[1]
Ligand Pharmaceut Inc, San Diego, CA 92121 USA
来源
:
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM
|
1999年
/ 84卷
/ 10期
关键词
:
D O I
:
10.1210/jc.84.10.3459
中图分类号
:
R5 [内科学];
学科分类号
:
1002 ;
100201 ;
摘要
:
引用
收藏
页码:3459 / 3462
页数:4
相关论文
共 27 条
[21]
Identification characterization, and tissue distribution of human peroxisome proliferator-activated receptor (PPAR) isoforms PPAR gamma 2 versus PPAR gamma 1 and activation with retinoid X receptor agonists and antagonists
[J].
Mukherjee, R
论文数:
0
引用数:
0
h-index:
0
机构:
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
Mukherjee, R
;
Jow, L
论文数:
0
引用数:
0
h-index:
0
机构:
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
Jow, L
;
Croston, GE
论文数:
0
引用数:
0
h-index:
0
机构:
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
Croston, GE
;
Paterniti, JR
论文数:
0
引用数:
0
h-index:
0
机构:
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
Paterniti, JR
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
1997,
272
(12)
:8071
-8076
[22]
Nieschlag E., 1998, TESTOSTERONE, P293, DOI [10.1007/978-3-642-72185-4_10, DOI 10.1007/978-3-642-72185-4_10]
[23]
OSTEOPOROSIS IN MEN
[J].
ORWOLL, ES
论文数:
0
引用数:
0
h-index:
0
机构:
OREGON HLTH SCI UNIV, PORTLAND, OR 97207 USA
OREGON HLTH SCI UNIV, PORTLAND, OR 97207 USA
ORWOLL, ES
;
KLEIN, RF
论文数:
0
引用数:
0
h-index:
0
机构:
OREGON HLTH SCI UNIV, PORTLAND, OR 97207 USA
OREGON HLTH SCI UNIV, PORTLAND, OR 97207 USA
KLEIN, RF
.
ENDOCRINE REVIEWS,
1995,
16
(01)
:87
-116
[24]
Transactivation by retinoid X receptor peroxisome proliferator-activated receptor γ (PPARγ) heterodimers:: Intermolecular synergy requires only the PPARγ hormone-dependent activation function
[J].
Schulman, IG
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Schulman, IG
;
Shao, G
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Shao, G
;
Heyman, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Heyman, RA
.
MOLECULAR AND CELLULAR BIOLOGY,
1998,
18
(06)
:3483
-3494
[25]
Effect of testosterone treatment on bone mineral density in men over 65 years of age
[J].
Snyder, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Snyder, PJ
;
Peachey, H
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Peachey, H
;
Hannoush, P
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Hannoush, P
;
Berlin, JA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Berlin, JA
;
Loh, L
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Loh, L
;
Holmes, JH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Holmes, JH
;
Dlewati, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Dlewati, A
;
Staley, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Staley, J
;
Santanna, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Santanna, J
;
Kapoor, SC
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Kapoor, SC
;
Attie, MF
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Attie, MF
;
Haddad, JG
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Haddad, JG
;
Strom, BL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Strom, BL
.
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM,
1999,
84
(06)
:1966
-1972
[26]
5-aryl-1,2-dihydrochromeno[3,4-f]quinolines: A novel class of nonsteroidal human progesterone receptor agonists
[J].
Zhi, L
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Zhi, L
;
Tegley, CM
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Tegley, CM
;
Kallel, EA
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Kallel, EA
;
Marschke, KB
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Marschke, KB
;
Mais, DE
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Mais, DE
;
Gottardis, MM
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Gottardis, MM
;
Jones, TK
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Jones, TK
.
JOURNAL OF MEDICINAL CHEMISTRY,
1998,
41
(03)
:291
-302
[27]
Switching androgen receptor antagonists to agonists by modifying C-ring substituents on piperidino[3,2-g]quinolinone
[J].
Zhi, L
论文数:
0
引用数:
0
h-index:
0
机构:
Dept Med Chem, San Diego, CA 92121 USA
Zhi, L
;
Tegley, CM
论文数:
0
引用数:
0
h-index:
0
机构:
Dept Med Chem, San Diego, CA 92121 USA
Tegley, CM
;
Marschke, KB
论文数:
0
引用数:
0
h-index:
0
机构:
Dept Med Chem, San Diego, CA 92121 USA
Marschke, KB
;
Jones, TK
论文数:
0
引用数:
0
h-index:
0
机构:
Dept Med Chem, San Diego, CA 92121 USA
Jones, TK
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1999,
9
(07)
:1009
-1012
←
1
2
3
→
共 27 条
[21]
Identification characterization, and tissue distribution of human peroxisome proliferator-activated receptor (PPAR) isoforms PPAR gamma 2 versus PPAR gamma 1 and activation with retinoid X receptor agonists and antagonists
[J].
Mukherjee, R
论文数:
0
引用数:
0
h-index:
0
机构:
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
Mukherjee, R
;
Jow, L
论文数:
0
引用数:
0
h-index:
0
机构:
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
Jow, L
;
Croston, GE
论文数:
0
引用数:
0
h-index:
0
机构:
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
Croston, GE
;
Paterniti, JR
论文数:
0
引用数:
0
h-index:
0
机构:
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
LIGAND PHARMACEUT INC,DEPT NEW LEADS DISCOVERY,SAN DIEGO,CA 92121
Paterniti, JR
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
1997,
272
(12)
:8071
-8076
[22]
Nieschlag E., 1998, TESTOSTERONE, P293, DOI [10.1007/978-3-642-72185-4_10, DOI 10.1007/978-3-642-72185-4_10]
[23]
OSTEOPOROSIS IN MEN
[J].
ORWOLL, ES
论文数:
0
引用数:
0
h-index:
0
机构:
OREGON HLTH SCI UNIV, PORTLAND, OR 97207 USA
OREGON HLTH SCI UNIV, PORTLAND, OR 97207 USA
ORWOLL, ES
;
KLEIN, RF
论文数:
0
引用数:
0
h-index:
0
机构:
OREGON HLTH SCI UNIV, PORTLAND, OR 97207 USA
OREGON HLTH SCI UNIV, PORTLAND, OR 97207 USA
KLEIN, RF
.
ENDOCRINE REVIEWS,
1995,
16
(01)
:87
-116
[24]
Transactivation by retinoid X receptor peroxisome proliferator-activated receptor γ (PPARγ) heterodimers:: Intermolecular synergy requires only the PPARγ hormone-dependent activation function
[J].
Schulman, IG
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Schulman, IG
;
Shao, G
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Shao, G
;
Heyman, RA
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Ligand Pharmaceut Inc, Dept Retinoid Res, San Diego, CA 92121 USA
Heyman, RA
.
MOLECULAR AND CELLULAR BIOLOGY,
1998,
18
(06)
:3483
-3494
[25]
Effect of testosterone treatment on bone mineral density in men over 65 years of age
[J].
Snyder, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Snyder, PJ
;
Peachey, H
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Peachey, H
;
Hannoush, P
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Hannoush, P
;
Berlin, JA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Berlin, JA
;
Loh, L
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Loh, L
;
Holmes, JH
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Holmes, JH
;
Dlewati, A
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Dlewati, A
;
Staley, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Staley, J
;
Santanna, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Santanna, J
;
Kapoor, SC
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Kapoor, SC
;
Attie, MF
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Attie, MF
;
Haddad, JG
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Haddad, JG
;
Strom, BL
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Penn, Sch Med, Dept Med, Philadelphia, PA 19104 USA
Strom, BL
.
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM,
1999,
84
(06)
:1966
-1972
[26]
5-aryl-1,2-dihydrochromeno[3,4-f]quinolines: A novel class of nonsteroidal human progesterone receptor agonists
[J].
Zhi, L
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Zhi, L
;
Tegley, CM
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Tegley, CM
;
Kallel, EA
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Kallel, EA
;
Marschke, KB
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Marschke, KB
;
Mais, DE
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Mais, DE
;
Gottardis, MM
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Gottardis, MM
;
Jones, TK
论文数:
0
引用数:
0
h-index:
0
机构:
Ligand Pharmaceut Inc, Dept Med Chem, San Diego, CA 92121 USA
Jones, TK
.
JOURNAL OF MEDICINAL CHEMISTRY,
1998,
41
(03)
:291
-302
[27]
Switching androgen receptor antagonists to agonists by modifying C-ring substituents on piperidino[3,2-g]quinolinone
[J].
Zhi, L
论文数:
0
引用数:
0
h-index:
0
机构:
Dept Med Chem, San Diego, CA 92121 USA
Zhi, L
;
Tegley, CM
论文数:
0
引用数:
0
h-index:
0
机构:
Dept Med Chem, San Diego, CA 92121 USA
Tegley, CM
;
Marschke, KB
论文数:
0
引用数:
0
h-index:
0
机构:
Dept Med Chem, San Diego, CA 92121 USA
Marschke, KB
;
Jones, TK
论文数:
0
引用数:
0
h-index:
0
机构:
Dept Med Chem, San Diego, CA 92121 USA
Jones, TK
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1999,
9
(07)
:1009
-1012
←
1
2
3
→