The use of solubility parameters in pharmaceutical dosage form design

被引：244

作者：

Hancock, BC

York, P

Rowe, RC

机构：

[1] UNIV BRADFORD,SCH PHARM,BRADFORD BD7 1DP,W YORKSHIRE,ENGLAND

[2] ZENECA PHARMACEUT,MACCLESFIELD,CHESHIRE,ENGLAND

来源：

INTERNATIONAL JOURNAL OF PHARMACEUTICS | 1997年 / 148卷 / 01期

关键词：

cohesive energy density; solubility parameter; interaction; polarity; formulation;

D O I：

10.1016/S0378-5173(96)04828-4

中图分类号：

R9 [药学];

学科分类号：

1007 ;

摘要：

The use and potential of solubility parameters for pharmaceutical dosage form design are reviewed in this paper. Specific reference is given to the development of the approach, its previous usage and likely future applications. The advantages, assumptions and limitations of this type of approach are also described. (C) 1997 Elsevier Science B.V.

引用

页码：1 / 21

页数：21

共 109 条

[1] EXTENDED HILDEBRAND APPROACH - SOLUBILITY OF CAFFEINE IN DIOXANE-WATER MIXTURES [J].

ADJEI, A ;

NEWBURGER, J ;

MARTIN, A .

JOURNAL OF PHARMACEUTICAL SCIENCES, 1980, 69 (06) :659-661

[2] THE MOLECULAR-BASIS OF MOISTURE EFFECTS ON THE PHYSICAL AND CHEMICAL-STABILITY OF DRUGS IN THE SOLID-STATE [J].

AHLNECK, C ;

ZOGRAFI, G .

INTERNATIONAL JOURNAL OF PHARMACEUTICS, 1990, 62 (2-3) :87-95

[3]

[Anonymous], INT J PHARM

[4]

[Anonymous], J PHARM SCI

[5] HANSEN SOLUBILITY PARAMETERS FOR SELECTED CELLULOSE ETHER DERIVATIVES AND THEIR USE IN THE PHARMACEUTICAL-INDUSTRY [J].

ARCHER, WL .

DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY, 1992, 18 (05) :599-616

[6]

Bajpai AK, 1996, REV ROUM CHIM, V41, P219

[7] SOLVENT SELECTIVITY IN REVERSED-PHASE HIGH-PRESSURE LIQUID-CHROMATOGRAPHY [J].

BAKALYAR, SR ;

MCILWRICK, R ;

ROGGENDORF, E .

JOURNAL OF CHROMATOGRAPHY, 1977, 142 (NOV) :353-365

[8] Influence of surface free energies and cohesion parameters on pharmaceutical material interaction parameters-theoretical simulations [J].

Barra, J ;

Lescure, F ;

Doelker, E .

PHARMACEUTICAL RESEARCH, 1996, 13 (11) :1746-1751

[9]

Barton A.F. M., 1991, Handbook of Solubility Parameters and Other Cohesion Parameters, V2nd

[10] APPLICATIONS OF SOLUBILITY PARAMETERS AND OTHER COHESION PARAMETERS IN POLYMER SCIENCE AND TECHNOLOGY [J].

BARTON, AFM .

PURE AND APPLIED CHEMISTRY, 1985, 57 (07) :905-912

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