Facile construction of functionalized 4H-chromene via tandem benzylation and cyclization

被引:82
作者
Fan, Jinmin
Wang, Zhiyong [1 ]
机构
[1] Univ Sci & Technol China, Joint Lab Green Synthet Chem, Hefei Natl Lab Phys Sci Microscale, Hefei 230026, Peoples R China
基金
中国国家自然科学基金;
关键词
D O I
10.1039/b812046c
中图分类号
O6 [化学];
学科分类号
0703 [化学];
摘要
A series of functionalized 4H-chromenes have been constructed by using a novel FeCl3-catalyzed benzylation-cyclization tandem reaction.
引用
收藏
页码:5381 / 5383
页数:3
相关论文
共 29 条
[1]
Domino reactions of 1,3-bis-silyl enol ethers with benzopyrylium triflates:: Efficient synthesis of fluorescent 6H-benzo[c]chromen-6-ones, dibenzo[c,d]chromen-6-ones, and 2,3-dihydro-1H-4,6-dioxachrysen-5-ones [J].
Appel, B ;
Saleh, NNR ;
Langer, P .
CHEMISTRY-A EUROPEAN JOURNAL, 2006, 12 (04) :1221-1236
[2]
ANTIINFLAMMATORY MECHANISM OF CORDIACHROMENE-A ACTION [J].
BENSLIMANE, AF ;
POUCHUS, YF ;
VERBIST, JF ;
PETIT, JY ;
BRION, JD ;
WELIN, L .
JOURNAL OF CLINICAL PHARMACOLOGY, 1995, 35 (03) :298-301
[3]
ENANTIOSELECTIVE TOTAL SYNTHESIS OF MIROESTROL [J].
COREY, EJ ;
WU, LI .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1993, 115 (20) :9327-9328
[4]
Rhodomyrtone, an antibiotic from Rhodomyrtus tomentosa [J].
Dachriyanus ;
Salni ;
Sargent, MV ;
Skelton, BW ;
Soediro, I ;
Sutisna, M ;
White, AH ;
Yulinah, E .
AUSTRALIAN JOURNAL OF CHEMISTRY, 2002, 55 (03) :229-232
[5]
O-arylation versus C-arylation: Copper-catalyzed intramolecular coupling of aryl bromides with 1,3-dicarbonyls [J].
Fang, Yewen ;
Li, Chaozhong .
JOURNAL OF ORGANIC CHEMISTRY, 2006, 71 (17) :6427-6431
[6]
Reactions of salicyl N-tosylimines or salicylaldehydes with diethyl acetylenedicarboxylate for the synthesis of highly functionalized chromenes [J].
Guo, Ying-Wen ;
Shi, Yong-Ling ;
Li, Hong-Bin ;
Shi, Min .
TETRAHEDRON, 2006, 62 (25) :5875-5882
[7]
Discovery of potent chromen-4-one inhibitors of the DNA-dependent protein kinase (DNA-PK) using a small-molecule library approach [J].
Hardcastle, IR ;
Cockcroft, X ;
Curtin, NJ ;
El-Murr, MD ;
Leahy, JJJ ;
Stockley, M ;
Golding, BT ;
Rigoreau, L ;
Richardson, C ;
Smith, GCM ;
Griffin, RJ .
JOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (24) :7829-7846
[8]
An efficient and general iron-catalyzed arylation of benzyl alcohols and benzyl carboxylates [J].
Iovel, I ;
Mertins, K ;
Kischel, J ;
Zapf, A ;
Beller, M .
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2005, 44 (25) :3913-3917
[9]
Aqua mediated synthesis of substituted 2-amino-4H-chromenes and in vitro study as antibacterial agents [J].
Kidwai, M ;
Saxena, S ;
Khan, MKR ;
Thukral, SS .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (19) :4295-4298
[10]
A general and efficient iron-catalyzed benzylation of 1,3-dicarbonyl compounds [J].
Kischel, Jette ;
Mertins, Kristin ;
Michalik, Dirk ;
Zapf, Alexander ;
Beller, Matthias .
ADVANCED SYNTHESIS & CATALYSIS, 2007, 349 (06) :865-870