Microwave-assisted synthesis utilizing supported reagents: a rapid and versatile synthesis of 1,5-diarylpyrazoles

被引：37

作者：

Humphries, PS ^{[1
]}

Finefield, JM ^{[1
]}

机构：

[1] Pfizer Global R&D, Dept Med Chem, San Diego, CA 92121 USA

来源：

TETRAHEDRON LETTERS | 2006年 / 47卷 / 14期

关键词：

D O I：

10.1016/j.tetlet.2006.01.100

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The application of microwave heating to a silica-assisted solution-phase synthesis technique has been utilized to develop a rapid and efficient two-step protocol for the preparation of pyrazoles from aryl methyl ketone and aryl hydrazine monomers. (c) 2006 Elsevier Ltd. All rights reserved.

引用

页码：2443 / 2446

页数：4

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