共 30 条
[1]
Hit generation and exploration:: Imidazo[4,5-b] pyridine derivatives as inhibitors of Aurora kinases
[J].
Bavetsias, Vassilios
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Sun, Chongbo
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Bouloc, Nathalie
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Reynisson, Johannes
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Workman, Paul
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Linardopoulos, Spiros
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McDonald, Edward
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BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2007, 17 (23)
:6567-6571

Bavetsias, Vassilios
论文数: 0 引用数: 0
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机构:
Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England

Sun, Chongbo
论文数: 0 引用数: 0
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机构:
Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England

Bouloc, Nathalie
论文数: 0 引用数: 0
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机构:
Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England

Reynisson, Johannes
论文数: 0 引用数: 0
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机构:
Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England

Workman, Paul
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England

Linardopoulos, Spiros
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England

McDonald, Edward
论文数: 0 引用数: 0
h-index: 0
机构:
Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England Inst Canc Res, Canc Res UK Lab, Canc Res UK Ctr Canc Therapeut, Dept Chem, Sutton SM2 5NG, Surrey, England
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The Protein Data Bank
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NUCLEIC ACIDS RESEARCH,
2000, 28 (01)
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Berman, HM
论文数: 0 引用数: 0
h-index: 0
机构: Rutgers State Univ, Dept Chem, Piscataway, NJ 08854 USA

Westbrook, J
论文数: 0 引用数: 0
h-index: 0
机构: Rutgers State Univ, Dept Chem, Piscataway, NJ 08854 USA

Feng, Z
论文数: 0 引用数: 0
h-index: 0
机构: Rutgers State Univ, Dept Chem, Piscataway, NJ 08854 USA

Gilliland, G
论文数: 0 引用数: 0
h-index: 0
机构: Rutgers State Univ, Dept Chem, Piscataway, NJ 08854 USA

Bhat, TN
论文数: 0 引用数: 0
h-index: 0
机构: Rutgers State Univ, Dept Chem, Piscataway, NJ 08854 USA

Weissig, H
论文数: 0 引用数: 0
h-index: 0
机构: Rutgers State Univ, Dept Chem, Piscataway, NJ 08854 USA

Shindyalov, IN
论文数: 0 引用数: 0
h-index: 0
机构: Rutgers State Univ, Dept Chem, Piscataway, NJ 08854 USA

Bourne, PE
论文数: 0 引用数: 0
h-index: 0
机构: Rutgers State Univ, Dept Chem, Piscataway, NJ 08854 USA
[3]
A homologue of Drosophila aurora kinase is oncogenic and amplified in human colorectal cancers
[J].
Bischoff, JR
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Anderson, L
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Zhu, YF
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Mossie, K
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Ng, L
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Souza, B
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Schryver, B
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Flanagan, P
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Clairvoyant, F
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Ginther, C
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Novotny, M
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Plowman, GD
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EMBO JOURNAL,
1998, 17 (11)
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Bischoff, JR
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Anderson, L
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Zhu, YF
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h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Mossie, K
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Ng, L
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Souza, B
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h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Schryver, B
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Flanagan, P
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Clairvoyant, F
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Ginther, C
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h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Chan, CSM
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Novotny, M
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Slamon, DJ
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA

Plowman, GD
论文数: 0 引用数: 0
h-index: 0
机构: SUGEN Inc, Redwood City, CA 94063 USA
[4]
CHARMM - A PROGRAM FOR MACROMOLECULAR ENERGY, MINIMIZATION, AND DYNAMICS CALCULATIONS
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BROOKS, BR
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BRUCCOLERI, RE
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OLAFSON, BD
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STATES, DJ
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SWAMINATHAN, S
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KARPLUS, M
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JOURNAL OF COMPUTATIONAL CHEMISTRY,
1983, 4 (02)
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BROOKS, BR
论文数: 0 引用数: 0
h-index: 0

BRUCCOLERI, RE
论文数: 0 引用数: 0
h-index: 0

OLAFSON, BD
论文数: 0 引用数: 0
h-index: 0

STATES, DJ
论文数: 0 引用数: 0
h-index: 0

SWAMINATHAN, S
论文数: 0 引用数: 0
h-index: 0

KARPLUS, M
论文数: 0 引用数: 0
h-index: 0
[5]
Aurora kinases: New targets for cancer therapy
[J].
Carvajal, Richard D.
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Tse, Archie
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Schwartz, Gary K.
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CLINICAL CANCER RESEARCH,
2006, 12 (23)
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Carvajal, Richard D.
论文数: 0 引用数: 0
h-index: 0
机构: Mem Sloan Kettering Canc Ctr, Dept Med, Melanoma Sarcoma Serv, New York, NY 10021 USA

Tse, Archie
论文数: 0 引用数: 0
h-index: 0
机构: Mem Sloan Kettering Canc Ctr, Dept Med, Melanoma Sarcoma Serv, New York, NY 10021 USA

Schwartz, Gary K.
论文数: 0 引用数: 0
h-index: 0
机构: Mem Sloan Kettering Canc Ctr, Dept Med, Melanoma Sarcoma Serv, New York, NY 10021 USA
[6]
Cee V. J., 2007, [No title captured], Patent No. [07087276, WO07087276]
[7]
Aurora A, meiosis and mitosis
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Crane, R
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Gadea, B
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Littlepage, L
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Wu, H
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Ruderman, JV
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BIOLOGY OF THE CELL,
2004, 96 (03)
:215-229

论文数: 引用数:
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机构:

Gadea, B
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dept Cell Biol, Boston, MA 02115 USA Harvard Univ, Sch Med, Dept Cell Biol, Boston, MA 02115 USA

Littlepage, L
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dept Cell Biol, Boston, MA 02115 USA Harvard Univ, Sch Med, Dept Cell Biol, Boston, MA 02115 USA

Wu, H
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dept Cell Biol, Boston, MA 02115 USA Harvard Univ, Sch Med, Dept Cell Biol, Boston, MA 02115 USA

Ruderman, JV
论文数: 0 引用数: 0
h-index: 0
机构:
Harvard Univ, Sch Med, Dept Cell Biol, Boston, MA 02115 USA Harvard Univ, Sch Med, Dept Cell Biol, Boston, MA 02115 USA
[8]
Potent and selective aurora inhibitors identified by the expansion of a novel scaffold for protein kinase inhibition
[J].
Fancelli, D
;
Berta, D
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Bindi, S
;
Cameron, A
;
Cappella, P
;
Carpinelli, P
;
Catana, C
;
Forte, B
;
Giordano, P
;
Giorgini, ML
;
Mantegani, S
;
Marsiglio, A
;
Meroni, M
;
Moll, J
;
Pittalà, V
;
Roletto, F
;
Severino, D
;
Soncini, C
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Storici, P
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Tonani, R
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Varasi, M
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Vulpetti, A
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Vianello, P
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JOURNAL OF MEDICINAL CHEMISTRY,
2005, 48 (08)
:3080-3084

Fancelli, D
论文数: 0 引用数: 0
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Berta, D
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Bindi, S
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Cameron, A
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Cappella, P
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Carpinelli, P
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Catana, C
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Forte, B
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Giordano, P
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Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Giorgini, ML
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Mantegani, S
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Marsiglio, A
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Meroni, M
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Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Moll, J
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Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Pittalà, V
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Roletto, F
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Severino, D
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Soncini, C
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Storici, P
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Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Tonani, R
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Varasi, M
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Vulpetti, A
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Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy

Vianello, P
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机构:
Nerviano Med Sci Oncol, I-20014 Milan, Italy Nerviano Med Sci Oncol, I-20014 Milan, Italy
[9]
1,4,5,6-tetrahydropyrrolo[3,4-c] pyrazoles:: Identification of a potent aurora kinase inhibitor with a favorable antitumor kinase inhibition profile
[J].
Fancelli, Daniele
;
Moll, Jurgen
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Varasi, Mario
;
Bravo, Rodrigo
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Artico, Roberta
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Berta, Daniela
;
Bindi, Simona
;
Cameron, Alexander
;
Candiani, Ilaria
;
Cappella, Paolo
;
Carpinelli, Patrizia
;
Croci, Walter
;
Forte, Barbara
;
Giorgini, Maria Laura
;
Klapwijk, Jan
;
Marsiglio, Aurelio
;
Pesenti, Enrico
;
Rocchetti, Maurizio
;
Roletto, Fulvia
;
Severino, Dino
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Soncini, Chiara
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Storici, Paola
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Tonani, Roberto
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Zugnoni, Paola
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Vianello, Paola
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JOURNAL OF MEDICINAL CHEMISTRY,
2006, 49 (24)
:7247-7251

Fancelli, Daniele
论文数: 0 引用数: 0
h-index: 0
机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Moll, Jurgen
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Varasi, Mario
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Bravo, Rodrigo
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Artico, Roberta
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Berta, Daniela
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Bindi, Simona
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Cameron, Alexander
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Candiani, Ilaria
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Cappella, Paolo
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Carpinelli, Patrizia
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Croci, Walter
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Forte, Barbara
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Giorgini, Maria Laura
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Klapwijk, Jan
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Marsiglio, Aurelio
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Pesenti, Enrico
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Rocchetti, Maurizio
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Roletto, Fulvia
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Severino, Dino
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Soncini, Chiara
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Storici, Paola
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Tonani, Roberto
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Zugnoni, Paola
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Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy

Vianello, Paola
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机构:
Nerviano Med Sci SrL, I-20014 Milan, Italy Nerviano Med Sci SrL, I-20014 Milan, Italy
[10]
Proteomic characterization of the angiogenesis inhibitor SU6668 reveals multiple impacts on cellular kinase signaling
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Godl, K
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Gruss, OJ
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Eickhoff, J
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Wissing, J
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Blencke, S
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Degen, H
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Brehmer, D
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Horváth, Z
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Kéri, G
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Ullrich, A
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Daub, H
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CANCER RESEARCH,
2005, 65 (15)
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Godl, K
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h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Gruss, OJ
论文数: 0 引用数: 0
h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Eickhoff, J
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机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Wissing, J
论文数: 0 引用数: 0
h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Blencke, S
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机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Weber, M
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机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Degen, H
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机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Brehmer, D
论文数: 0 引用数: 0
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机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Orfi, L
论文数: 0 引用数: 0
h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Horváth, Z
论文数: 0 引用数: 0
h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Kéri, G
论文数: 0 引用数: 0
h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Müller, S
论文数: 0 引用数: 0
h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Cotten, M
论文数: 0 引用数: 0
h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Ullrich, A
论文数: 0 引用数: 0
h-index: 0
机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany

Daub, H
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机构: Max Planck Inst Biochem, Dept Biol Mol, D-82152 Martinsried, Germany