Asymmetric synthesis of α-fluoro ketones using α-fluoro oxazolidinone carboximides

被引：72

作者：

Davis, FA ^{[1
]}

Kasu, PVN ^{[1
]}

机构：

[1] Temple Univ, Dept Chem, Philadelphia, PA 19122 USA

来源：

TETRAHEDRON LETTERS | 1998年 / 39卷 / 34期

关键词：

D O I：

10.1016/S0040-4039(98)01296-9

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Addition of Grignard reagents io enantiopure alpha-fluoro N-methoxy-N-methylamides 5 affords alpha-fluoro ketones (R)-6 in >96% ee. (C) 1998 Elsevier Science Ltd. All rights reserved.

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收藏

页码：6135 / 6138

页数：4

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