The design and synthesis of novel 3-[2-indol-1-yl-ethyl]-1-H-indole derivatives as selective inhibitors of CDK4

被引：54

作者：

Aubry, C

Patel, A

Mahale, S

Chaudhuri, B

Maréchal, JD

Suteliffe, MJ

Jenkins, PR ^{[1
]}

机构：

[1] Univ Leicester, Dept Chem, Leicester LE1 7RH, Leics, England

[2] De Montfort Univ, Leicester Sch Pharm, Leicester LE1 9BH, Leics, England

[3] Univ Leicester, Dept Biochem & Chem, Leicester LE1 7RH, Leics, England

来源：

TETRAHEDRON LETTERS | 2005年 / 46卷 / 09期

关键词：

indole; CDK4; fascaplysin; 3-[2-indol-l-yl-ethyl]-1H-indole; molecular modelling; IC50;

D O I：

10.1016/j.tetlet.2005.01.054

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1423 / 1425

页数：3

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