Investigation of new potent KDO-8-phosphate synthetase inhibitors

被引：21

作者：

Coutrot, P

Dumarçay, S

Finance, C

Tabyaoui, M

Tabyaoui, B

Grison, C

机构：

[1] UHP, Inst Nanceien Chim Mol, Lab Chim Organ 2, F-54506 Vandoeuvre Nancy, France

[2] UHP, GEVSM, CNRS, Inst Nanceien Chim Mol, F-54506 Vandoeuvre Nancy, France

[3] Univ Chouaib Doukkali, Fac Sci, Dept Chim, El Jadida, Morocco

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1999年 / 9卷 / 07期

关键词：

D O I：

10.1016/S0960-894X(99)00111-0

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A total synthesis of (Z,E)-D-Glucophosphoenolpyruvate and its carboxylic ester derivatives is described in four or five steps from 2,3 : 5,6-Di-O-isopropylidene-4-O-t-butyldimethylsilyl-D-glucose (C) 1999 Elsevier Science Ltd. All rights reserved.

引用

页码：949 / 952

页数：4

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