Antithrombotics serine proteases

被引:70
作者
Ripka, WC
Vlasuk, GP
机构
[1] Corvas International, San Diego
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 32 | 1997年 / 32卷
关键词
D O I
10.1016/S0065-7743(08)61466-9
中图分类号
O69 [应用化学];
学科分类号
081704 ;
摘要
[No abstract available]
引用
收藏
页码:71 / 89
页数:19
相关论文
共 114 条
[41]   GUIDE TO ANTICOAGULANT-THERAPY .2. ORAL ANTICOAGULANTS [J].
HIRSH, J ;
FUSTER, V .
CIRCULATION, 1994, 89 (03) :1469-1480
[42]   HEPARINS [J].
HIRSH, J .
FIBRINOLYSIS, 1995, 9 :66-68
[43]  
HOYLE W, 1996, Patent No. 9629327
[44]   Derivatives of 5-amidine indole as inhibitors of thrombin catalytic activity [J].
Iwanowicz, EJ ;
Lau, WF ;
Lin, J ;
Roberts, DGM ;
Seiler, SM .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1996, 6 (12) :1339-1344
[45]   RETRO-BINDING TRIPEPTIDE THROMBIN ACTIVE-SITE INHIBITORS - DISCOVERY, SYNTHESIS, AND MOLECULAR MODELING [J].
IWANOWICZ, EJ ;
LAU, WF ;
LIN, J ;
ROBERTS, DGM ;
SELLERS, SM .
JOURNAL OF MEDICINAL CHEMISTRY, 1994, 37 (14) :2122-2124
[46]   INFLUENCE OF BLOCKADE AT SPECIFIC LEVELS OF THE COAGULATION CASCADE ON RESTENOSIS IN A RABBIT ATHEROSCLEROTIC FEMORAL-ARTERY INJURY MODEL [J].
JANG, YS ;
GUZMAN, LA ;
LINCOFF, AM ;
GOTTSAUNERWOLF, M ;
FORUDI, F ;
HART, CE ;
COURTMAN, DW ;
EZBAN, M ;
ELLIS, SG ;
TOPOL, EJ .
CIRCULATION, 1995, 92 (10) :3041-3050
[47]  
KAISER B, 1985, BIOMED BIOCHIM ACTA, V44, P1201
[48]   Factor V-Leiden and thrombophilia [J].
Kalafatis, M ;
Mann, KG .
ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY, 1997, 17 (04) :620-627
[49]   A soluble tissue factor mutant is a selective anticoagulant and antithrombotic agent [J].
Kelley, RF ;
Refino, CJ ;
OConnell, MP ;
Modi, N ;
Sehl, P ;
Lowe, D ;
Pater, C ;
Bunting, S .
BLOOD, 1997, 89 (09) :3219-3227
[50]  
KIM KS, 1996, MED CHEM RES, P377