Progress in Structure Based Drug Design for G Protein-Coupled Receptors

被引：157

作者：

Congreve, Miles ^{[1
]}

Langmead, Christopher J. ^{[1
]}

Mason, Jonathan S. ^{[1
]}

Marshall, Fiona H. ^{[1
]}

机构：

[1] Heptares Therapeut Ltd, Welwyn Garden City AL7 3AX, Herts, England

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 2011年 / 54卷 / 13期

关键词：

SITE-DIRECTED MUTAGENESIS; X-RAY-STRUCTURE; CRYSTAL-STRUCTURE; BINDING-SITE; ALLOSTERIC MODULATION; PHARMACOLOGICAL CHARACTERIZATION; BETA(2)-ADRENERGIC RECEPTOR; ADENOSINE RECEPTORS; IN-SILICO; MOLECULAR RECOGNITION;

D O I：

10.1021/jm200371q

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：4283 / 4311

页数：29

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