Synthesis of anti-bacterial peptidomimetics derived from N-acylisatins

被引：26

作者：

Cheah, Wai Ching ^{[1
]}

Black, David StC ^{[1
]}

Goh, Wai Kean ^{[1
]}

Kumar, Naresh ^{[1
]}

机构：

[1] Univ New S Wales, Sch Chem, Sydney, NSW 2052, Australia

来源：

TETRAHEDRON LETTERS | 2008年 / 49卷 / 18期

基金：

澳大利亚研究理事会;

关键词：

D O I：

10.1016/j.tetlet.2008.03.007

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient synthetic strategy to mono- and bis-glyoxylamide derivatives via the reaction of N-acylisatins with a range of amino acids has been developed. Using this strategy, a series of new peptidomimetics have been synthesized. (c) 2008 Elsevier Ltd. All rights reserved.

引用

页码：2965 / 2968

页数：4

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