A practical protocol for the synthesis of 3-hydroxy-4,5-disubstituted pyridine derivatives from acyclic compounds

被引：14

作者：

Anastasia, L ^{[1
]}

Anastasia, M ^{[1
]}

Allevi, P ^{[1
]}

机构：

[1] Univ Milan, Dipartimento Chim & Biochim Med, I-20133 Milan, Italy

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 2001年 / 19期

关键词：

D O I：

10.1039/b105478n

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The paper reports a simple protocol for assembling a 3-hydroxy-4,5-disubstituted pyridine ring by reaction of allylamine or benzylamine and an alpha -bromo ketone and successive N-dealkylation.

引用

页码：2404 / 2408

页数：5

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