Morphan based substance P antagonists

被引：5

作者：

Cocker, JD

Davies, HG

机构：

[1] Department of Medicinal Chemistry I, Glaxo R. and D. Limited, Glaxo-Wellcome Medicines Res. Centre, Stevenage, Hertfordshire SG1 2NY, Gunnels Wood Road

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1996年 / 6卷 / 01期

关键词：

D O I：

10.1016/0960-894X(95)00552-5

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A bridged derivative of the substance P antagonist CP 99,994 has been prepared and shown to possess potent affinity for the NK1 receptor.

引用

页码：13 / 16

页数：4

共 10 条

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