One pot synthesis of unsymmetrically functionalized polyamines by a solid phase strategy starting from their symmetrical polyamine-counterparts.

被引：30

作者：

Byk, G

Frederic, M

Scherman, D

机构：

[1] UMR-133 Rhone-Poulenc Rorer Gencell, CNRS, 94403-Vitry sur Seine, 13

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 18期

关键词：

D O I：

10.1016/S0040-4039(97)00582-0

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

We have developed a solid phase methodology which allows a quick and easy access to a high number of mono-functionalized geometrically varied polyamines. The feasibility of the method was demonstrated by the unsymmetrical introduction of a single carboxylic acid functional group into differing symmetrical polyamines. (C) 1997 Elsevier Science Ltd.

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页码：3219 / 3222

页数：4

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