Lithium perchlorate-catalyzed three-component coupling:: A facile and general method for the synthesis of α-aminophosphonates under solvent-free conditions

被引:80
作者
Azizi, N [1 ]
Saidi, MR [1 ]
机构
[1] Sharif Univ Technol, Dept Chem, Tehran, Iran
关键词
D O I
10.1002/ejoc.200300479
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A simple, efficient, and general method has been developed for the synthesis of alpha-aminophosphonates in the presence of solid lithium perchlorate under solvent-free conditions. Thus secondary and tertiary alpha-aminophosphonates were synthesized relatively quickly in good yields at room temperature. ((C) Wiley-VCH Verlag GmbH & Co. KGaA, 69451 Weinheim, Germany, 2003).
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收藏
页码:4630 / 4633
页数:4
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