An efficient and mild CuI/L-proline-catalyzed arylation of acetylacetone or ethyl cyanoacetate

被引：78

作者：

Jiang, YW ^{[1
]}

Wu, N ^{[1
]}

Wu, HH ^{[1
]}

He, MY ^{[1
]}

机构：

[1] E China Normal Univ, Dept Chem, Shanghai Key Lab Green Chem & Chem Proc, Shanghai 200062, Peoples R China

来源：

SYNLETT | 2005年 / 18期

关键词：

cross coupling; arylation; aryl iodide; catalysis; additive;

D O I：

10.1055/s-2005-918921

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The coupling reaction of aryl iodides with acetylacetone or ethyl cyanoacetate under catalysis of CuI/L-proline works at relatively mild conditions to provide 3-aryl-2, 4-pentanediones and alpha-aryl cyanoacetates in moderate to good yields.

引用

页码：2731 / 2734

页数：4

共 45 条

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