Discovery and identification of lead compounds from combinatorial mixtures

被引:7
作者
Beutel, BA
机构
[1] Abbott Laboratories, IL 60064-3500, D-4PN AP10, Abbott Park
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 32 | 1997年 / 32卷
关键词
D O I
10.1016/S0065-7743(08)61484-0
中图分类号
O69 [应用化学];
学科分类号
081704 ;
摘要
[No abstract available]
引用
收藏
页码:261 / 268
页数:8
相关论文
共 43 条
[21]   COMBINATORIAL CHEMISTRY - DIRECT ANALYSIS OF BEAD SURFACE-ASSOCIATED MATERIALS [J].
HASKINS, NJ ;
HUNTER, DJ ;
ORGAN, AJ ;
RAHMAN, SS ;
THOM, C .
RAPID COMMUNICATIONS IN MASS SPECTROMETRY, 1995, 9 (14) :1437-1440
[22]   THE BROAD UTILITY OF SOLUBLE PEPTIDE LIBRARIES FOR DRUG DISCOVERY [J].
HOUGHTEN, RA .
GENE, 1993, 137 (01) :7-11
[23]   CREATION AND FUNCTIONAL SCREENING OF A MULTIUSE PEPTIDE LIBRARY [J].
JAYAWICKREME, CK ;
GRAMINSKI, GF ;
QUILLAN, JM ;
LERNER, MR .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1994, 91 (05) :1614-1618
[24]   ENCODED COMBINATORIAL PEPTIDE LIBRARIES CONTAINING NONNATURAL AMINO-ACIDS [J].
KERR, JM ;
BANVILLE, SC ;
ZUCKERMANN, RN .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1993, 115 (06) :2529-2531
[25]   Deconvolution of combinatorial libraries for drug discovery: Theoretical comparison of pooling strategies [J].
Konings, DAM ;
Wyatt, JR ;
Ecker, DJ ;
Freier, SM .
JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (14) :2710-2719
[26]   Synthetic library techniques: Subjective (biased and generic) thoughts and views [J].
Krchnak, V ;
Lebl, M .
MOLECULAR DIVERSITY, 1996, 1 (03) :193-216
[27]   Application of mass spectrometry for characterizing and identifying ligands from combinatorial libraries [J].
Loo, JA ;
DeJohn, DE ;
Loo, RRO ;
Andrews, PC .
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 31, 1996, 31 :319-325
[28]   GENERATION AND SCREENING OF AN OLIGONUCLEOTIDE-ENCODED SYNTHETIC PEPTIDE LIBRARY [J].
NEEDELS, MC ;
JONES, DG ;
TATE, EH ;
HEINKEL, GL ;
KOCHERSPERGER, LM ;
DOWER, WJ ;
BARRETT, RW ;
GALLOP, MA .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1993, 90 (22) :10700-10704
[29]   Versatile approach to encoding combinatorial organic syntheses using chemically robust secondary amine tags [J].
Ni, ZJ ;
Maclean, D ;
Holmes, CP ;
Murphy, MM ;
Ruhland, B ;
Jacobs, JW ;
Gordon, EM ;
Gallop, MA .
JOURNAL OF MEDICINAL CHEMISTRY, 1996, 39 (08) :1601-1608
[30]  
Ni ZJ, 1996, METHOD ENZYMOL, V267, P261