Trifluoromethylation of aryl and heteroaryl halides

[71] Organometallic chemistry of amidate complexes.: Accelerating effect of bidentate ligands on the reductive elimination of N-aryl amidates from palladium(II) [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2006, 128 (28) : 9044 - 9045

[72] Penta-substituted benzimidazoles as potent antagonists of the calcium-sensing receptor (CaSR-antagonists) [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (17) : 5161 - 5164

[73] Synthesis of α-trifluoromethylated nitrogen heterocycles [J]. JOURNAL OF ORGANIC CHEMISTRY, 2003, 68 (23) : 8932 - 8935

[74] GLAXO LTD, 2006, Patent No. 2006040192

[75] PREDICTIVE STRUCTURE-ACTIVITY-RELATIONSHIPS IN A SERIES OF PYRANOQUINOLINE DERIVATIVES - A NEW PRIMATE MODEL FOR THE IDENTIFICATION OF ANTIALLERGIC ACTIVITY [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (07) : 1445 - 1453

[76] Application of the Goldilocks Effect to the design of potent and selective inhibitors of phenylethanolamine N-methyltransferase:: Balancing pKa and steric effects in the optimization of 3-methyl-1,2,3,4-tetrahydroisoquinoline inhibitors by β-fluorination [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (10) : 2939 - 2952

[77] Inhibitors of phenylethanolamine N-methyltransferase devoid of α2-adrenoceptor affinity [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (23) : 5319 - 5323

[78] Facile Ar-CF3 bond formation at Pd.: Strikingly different outcomes of reductive elimination from [(Ph3P)2Pd(CF3)Ph] and [(Xantphos)Pd(CF3)Ph] [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2006, 128 (39) : 12644 - 12645

[79] The Organometallic Fluorine Chemistry of Palladium and Rhodium: Studies toward Aromatic Fluorination [J]. ACCOUNTS OF CHEMICAL RESEARCH, 2010, 43 (01) : 160 - 171

[80] Unexpected H2O-induced Ar-X activation with trifluoromethylpalladium(II) aryls [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2006, 128 (14) : 4632 - 4641

[71] Organometallic chemistry of amidate complexes.: Accelerating effect of bidentate ligands on the reductive elimination of N-aryl amidates from palladium(II) [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2006, 128 (28) : 9044 - 9045

[72] Penta-substituted benzimidazoles as potent antagonists of the calcium-sensing receptor (CaSR-antagonists) [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (17) : 5161 - 5164

[73] Synthesis of α-trifluoromethylated nitrogen heterocycles [J]. JOURNAL OF ORGANIC CHEMISTRY, 2003, 68 (23) : 8932 - 8935

[74] GLAXO LTD, 2006, Patent No. 2006040192

[75] PREDICTIVE STRUCTURE-ACTIVITY-RELATIONSHIPS IN A SERIES OF PYRANOQUINOLINE DERIVATIVES - A NEW PRIMATE MODEL FOR THE IDENTIFICATION OF ANTIALLERGIC ACTIVITY [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (07) : 1445 - 1453

[76] Application of the Goldilocks Effect to the design of potent and selective inhibitors of phenylethanolamine N-methyltransferase:: Balancing pKa and steric effects in the optimization of 3-methyl-1,2,3,4-tetrahydroisoquinoline inhibitors by β-fluorination [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (10) : 2939 - 2952

[77] Inhibitors of phenylethanolamine N-methyltransferase devoid of α2-adrenoceptor affinity [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (23) : 5319 - 5323

[78] Facile Ar-CF3 bond formation at Pd.: Strikingly different outcomes of reductive elimination from [(Ph3P)2Pd(CF3)Ph] and [(Xantphos)Pd(CF3)Ph] [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2006, 128 (39) : 12644 - 12645

[79] The Organometallic Fluorine Chemistry of Palladium and Rhodium: Studies toward Aromatic Fluorination [J]. ACCOUNTS OF CHEMICAL RESEARCH, 2010, 43 (01) : 160 - 171

[80] Unexpected H2O-induced Ar-X activation with trifluoromethylpalladium(II) aryls [J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2006, 128 (14) : 4632 - 4641