Trifluoromethylation of aryl and heteroaryl halides

被引：286

作者：

Roy, Sudipta ^{[1
]}

Gregg, Brian T. ^{[1
]}

Gribble, Gordon W. ^{[2
]}

Le, Van-Duc ^{[1
]}

Roy, Sujata ^{[1
]}

机构：

[1] AMRI, Dept Med Chem, 26 Corp Circle, Albany, NY 12212 USA

[2] Dartmouth Coll, Dept Chem, Hanover, NH 03755 USA

来源：

TETRAHEDRON | 2011年 / 67卷 / 12期

关键词：

CROSS-COUPLING REACTIONS; PHENYLETHANOLAMINE N-METHYLTRANSFERASE; FORMING REDUCTIVE ELIMINATION; ORGANIC FLUORINE-COMPOUNDS; NUCLEOPHILIC TRIFLUOROMETHYLATION; MEDICINAL CHEMISTRY; 1-AND 2-(TRIFLUOROMETHYL)NAPHTHALENES; BIOLOGICAL EVALUATION; SELECTIVE INHIBITORS; SYNTHETIC METHODS;

D O I：

10.1016/j.tet.2011.01.002

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

[No abstract available]

引用

页码：2161 / 2195

页数：35

共 212 条

[41] Copper-Mediated Oxidative Trifluoromethylation of Boronic Acids
Chu, Lingling
Qing, Feng-Ling
[J]. ORGANIC LETTERS, 2010, 12 (21) : 5060 - 5063
[42] CIDNUNEZ JM, 2009, Patent No. 20099033702
[43] CLAFFEY MM, 2007, Patent No. 2007034282
[44] THE TRIFLUOROMETHYLATION OF CHLOROAROMATICS USING THE COPPER-CF2BR2 - DIALKYLAMIDE REACTION SYSTEM
CLARK, JH
DENNESS, JE
MCCLINTON, MA
WYND, AJ
[J]. JOURNAL OF FLUORINE CHEMISTRY, 1990, 50 (03) : 411 - 426
[45] THE DIRECT TRIFLUOROMETHYLATION OF ARYL CHLORIDES USING BURTON REAGENT
CLARK, JH
MCCLINTON, MA
BLADE, RJ
[J]. JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1988, (10) : 638 - 639
[46] Clayton J., 2006, PCT Int. Appl., Patent No. [WO 2006/020879, 2006020879]
[47] Collins E.A., 2006, Patent No. 2006107784
[48] COMMONS TJ, 2008, Patent No. 200806099
[49] The metalation of 1-and 2-(trifluoromethyl)naphthalenes: noteworthy site selectivities
Cottet, F
Castagnetti, E
Schlosser, M
[J]. SYNTHESIS-STUTTGART, 2005, (05): : 798 - 803
[50] Logistic flexibility in the preparation of isomeric halopyridinecarboxylic acids
Cottet, F
Schlosser, M
[J]. TETRAHEDRON, 2004, 60 (51) : 11869 - 11874

← 1 2 3 4 5 6 7 8 9 10 →