GABAB receptor:: A new paradigm in G protein signaling

被引:229
作者
Couve, A
Moss, SJ
Pangalos, MN
机构
[1] SmithKline Beecham Pharmaceut, Neurosci Res, Harlow CM19 5AW, Essex, England
[2] UCL, MRC, Mol Cell Biol Lab, London WC1E 6BT, England
[3] UCL, Dept Pharmacol, London WC1E 6BT, England
关键词
D O I
10.1006/mcne.2000.0908
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
[No abstract available]
引用
收藏
页码:296 / 312
页数:17
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共 167 条
[51]   GAMMA-HYDROXYBUTYRIC ACID IN THE TREATMENT OF ALCOHOL DEPENDENCE - A DOUBLE-BLIND-STUDY [J].
GALLIMBERTI, L ;
FERRI, M ;
FERRARA, SD ;
FADDA, F ;
GESSA, GL .
ALCOHOLISM-CLINICAL AND EXPERIMENTAL RESEARCH, 1992, 16 (04) :673-676
[52]   Mutagenesis and modeling of the GABAB receptor extracellular domain support a Venus flytrap mechanism for ligand binding [J].
Galvez, T ;
Parmentier, ML ;
Joly, C ;
Malitschek, B ;
Kaupmann, K ;
Kuhn, R ;
Bittiger, H ;
Froestl, W ;
Bettler, B ;
Pin, JP .
JOURNAL OF BIOLOGICAL CHEMISTRY, 1999, 274 (19) :13362-13369
[53]   Ca2+ requirement for high-affinity γ-aminobutyric acid (GABA) binding at GABAB receptors:: Involvement of serine 269 of the GABABR1 subunit [J].
Galvez, T ;
Urwyler, S ;
Prézeu, L ;
Mosbacher, J ;
Joly, C ;
Malitschek, B ;
Heid, J ;
Brabet, I ;
Froestl, W ;
Bettler, B ;
Kaupmann, K ;
Pin, JP .
MOLECULAR PHARMACOLOGY, 2000, 57 (03) :419-426
[54]   The modulatory effects of high affinity GABAB receptor antagonists in an active avoidance learning paradigm in rats [J].
Getova, D ;
Bowery, NG .
PSYCHOPHARMACOLOGY, 1998, 137 (04) :369-373
[55]   Effects of GABA(B) receptor antagonists on learning and memory retention in a rat model of absence epilepsy [J].
Getova, D ;
Bowery, NG ;
Spassov, V .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1997, 320 (01) :9-13
[56]   Dopamine D1 and adenosine A1 receptors form functionally interacting heteromeric complexes [J].
Ginés, S ;
Hillion, J ;
Torvinen, M ;
Le Crom, S ;
Casadó, V ;
Canela, EI ;
Rondin, S ;
Lew, JY ;
Watson, S ;
Zoli, M ;
Agnati, LF ;
Vernier, P ;
Lluis, C ;
Ferré, S ;
Fuxe, K ;
Franco, R .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2000, 97 (15) :8606-8611
[57]   ENHANCEMENT OF MORPHINE ANALGESIA BY THE GABA(B) AGONIST BACLOFEN [J].
GORDON, NC ;
GEAR, RW ;
HELLER, PH ;
PAUL, S ;
MIASKOWSKI, C ;
LEVINE, JD .
NEUROSCIENCE, 1995, 69 (02) :345-349
[58]   Domain swapping in G-protein coupled receptor dimers [J].
Gouldson, PR ;
Snell, CR ;
Bywater, RP ;
Higgs, C ;
Reynolds, CA .
PROTEIN ENGINEERING, 1998, 11 (12) :1181-1193
[59]   HYPOTHERMIA INDUCED BY BACLOFEN, A POSSIBLE INDEX OF GABA-B RECEPTOR FUNCTION IN MICE, IS ENHANCED BY ANTIDEPRESSANT DRUGS AND ECS [J].
GRAY, JA ;
GOODWIN, GM ;
HEAL, DJ ;
GREEN, AR .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 92 (04) :863-870
[60]   INCREASED GABA-B RECEPTOR FUNCTION IN MOUSE FRONTAL-CORTEX AFTER REPEATED ADMINISTRATION OF ANTIDEPRESSANT DRUGS OR ELECTROCONVULSIVE SHOCKS [J].
GRAY, JA ;
GREEN, AR .
BRITISH JOURNAL OF PHARMACOLOGY, 1987, 92 (02) :357-362