Iron-catalyzed direct amination of azoles using formamides or amines as nitrogen sources in air

被引：133

作者：

Wang, Jian ^{[1
]}

Hou, Ji-Ting ^{[1
]}

Wen, Jun ^{[1
]}

Zhang, Ji ^{[1
]}

Yu, Xiao-Qi ^{[1
]}

机构：

[1] Sichuan Univ, Coll Chem, Minist Educ, Key Lab Green Chem & Technol, Chengdu 610064, Peoples R China

来源：

CHEMICAL COMMUNICATIONS | 2011年 / 47卷 / 12期

基金：

美国国家科学基金会;

关键词：

C-H BONDS; HYDROAMINATION; ALKENES; FUNCTIONALIZATION; ROUTE;

D O I：

10.1039/c0cc05811d

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A new iron-catalyzed, direct C-H amination of azoles at C2 has been developed by using formamides or amines as nitrogen sources. Imidazole is the only additive in the catalyst system and oxygen in air is employed during the transformation process.

引用

页码：3652 / 3654

页数：3

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